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61. 发明授权

US4357328A Heterocyclic substituted triazolyl phosphorous compounds and their use as insecticides 失效
标题翻译：杂环取代三唑基磷化合物及其作为杀虫剂的用途
公开(公告)号：US4357328A
公开(公告)日：1982-11-02
申请号：US260550
申请日：1981-05-04
申请人： Chester E. Pawloski
发明人： Chester E. Pawloski
IPC分类号： A01N57/08 , C07D213/77 , C07F9/6518 , C07F9/6558 , A01N57/16 , A01N57/24 , A01N57/32 , C07F9/65
CPC分类号： C07D213/77 , A01N57/08 , C07F9/65185 , C07F9/65583
摘要： Compounds are prepared which correspond to the formula ##STR1## wherein R represents a nitrogen containing heterocyclic radical corresponding to one of the formulae ##STR2## each X independently represents chloro, fluoro, bromo, nitro, alkyl of 1 to 4 carbon atoms, amino, mono- or dialkylamino wherein each alkyl group independently contains from 1 to 4 carbon atoms, alkoxy of 1 to 4 carbon atoms, alkylthio of 1 to 4 carbon atoms, alkylsulfinyl of 1 to 4 carbon atoms, alkylsulfonyl of 1 to 4 carbon atoms, cyano, trifluoromethyl, trichloromethyl, phenoxy or substituted phenoxy of the formula ##STR3## wherein each Z independently represents chloro, fluoro, bromo, nitro, cyano, alkoxy of 1 to 4 carbon atoms or alkylthio of 1 to 4 carbon atoms, with the proviso that when either n is 2 or 3, all X groups are sterically compatible with each other and all Z groups are sterically compatible with each other; Y represents oxygen or sulfur; each n can independently represent an integer of from 0 to 3, inclusive; R.sup.1 represents hydrogen, chloro, fluoro, bromo, alkyl of 1 to 4 carbon atoms, cycloalkyl of 3-6 carbon atoms, phenyl, phenylthio, alkoxy of 1 to 4 carbon atoms, alkylthio of 1 to 4 carbon atoms, alkylsulfinyl of 1 to 4 carbon atoms, alkylsulfonyl of 1 to 4 carbon atoms, thiocyanato, trifluoromethyl, trichloromethyl, amino, mono- or dialkylamino wherein each alkyl group independently contains from 1 to 4 carbon atoms; R.sup.2 represents methyl, ethyl, propyl or isobutyl and R.sup.3 represents methoxy, ethoxy, propoxy, ethyl, mono- or dialkylamino wherein each alkyl group independently contains from 1 to 4 carbon atoms, alkylthio of 1 to 4 carbon atoms or phenyl.
摘要翻译：制备符合下式的化合物：其中R表示与下式之一相对应的含氮杂环基：每个X独立地表示氯，氟，溴，硝基，1至4个碳原子的烷基，氨基，单 - 或二烷基氨基，其中每个烷基独立地含有1至4个碳原子，1至4个碳原子的烷氧基，1至4个碳原子的烷硫基，1个 1-4个碳原子的烷基磺酰基，氰基，三氟甲基，三氯甲基，苯氧基或取代的苯氧基，其中每个Z独立地表示氯，氟，溴，硝基，氰基，1-4个碳原子的烷氧基原子或1至4个碳原子的烷硫基，条件是当n为2或3时，所有X基彼此在空间上相容，所有Z基彼此空间相容; Y表示氧或硫; 每个n可以独立地表示0至3的整数，包括0和3; R 1表示氢，氯，氟，溴，1至4个碳原子的烷基，3-6个碳原子的环烷基，苯基，苯硫基，1至4个碳原子的烷氧基，1至4个碳原子的烷硫基，1至 4个碳原子，1至4个碳原子的烷基磺酰基，硫氰酸酯，三氟甲基，三氯甲基，氨基，一或二烷基氨基，其中每个烷基独立地含有1至4个碳原子; R 2表示甲基，乙基，丙基或异丁基，R 3表示甲氧基，乙氧基，丙氧基，乙基，单 - 或二烷基氨基，其中各烷基独立地含有1至4个碳原子，1至4个碳原子的烷硫基或苯基。

62. 发明授权

US4347251A Novel 3-substituted amino-1-substituted heteroaryl-2-pyrazolines 失效
标题翻译：新的3-取代的氨基-1-取代的杂芳基-2-吡唑啉
公开(公告)号：US4347251A
公开(公告)日：1982-08-31
申请号：US282827
申请日：1981-07-13
申请人： Joseph P. Joseph , John P. Dusza , Seymour Bernstein
发明人： Joseph P. Joseph , John P. Dusza , Seymour Bernstein
IPC分类号： C07C47/21 , C07D213/77 , C07D401/04 , A61K31/44
CPC分类号： C07D213/77 , C07C255/00 , C07C47/21
摘要： This disclosure describes novel 3-substituted amino-1-substituted heteroaryl-2-pyrazolines and their C.sub.4 and C.sub.5 analogs, effective as agents that ameliorate inflammation, analgesic agents, antibacterial agents and/or anti-fungal agents.
摘要翻译：本公开描述了新颖的3-取代的氨基-1-取代的杂芳基-2-吡唑啉及其C4和C5类似物，其有效作为改善炎症的药剂，止痛剂，抗菌剂和/或抗真菌剂。

63. 发明授权

US4298602A Heterocyclic substituted triazolyl phosphorous compounds and their use as insecticides 失效
标题翻译：杂环取代三唑基磷化合物及其作为杀虫剂的用途
公开(公告)号：US4298602A
公开(公告)日：1981-11-03
申请号：US084697
申请日：1979-10-15
申请人： Chester E. Pawloski
发明人： Chester E. Pawloski
IPC分类号： A01N57/08 , C07D213/77 , C07F9/6518 , C07F9/6558 , C07D213/02 , C07D215/02
CPC分类号： C07D213/77 , A01N57/08 , C07F9/65185 , C07F9/65583
摘要： Compounds are prepared which correspond to the formula ##STR1## wherein R represents a nitrogen containing heterocyclic radical corresponding to one of the formulae ##STR2## each X independently represents chloro, fluoro, bromo, nitro, alkyl of 1 to 4 carbon atoms, amino, mono- or dialkylamino wherein each alkyl group independently contains from 1 to 4 carbon atoms, alkoxy of 1 to 4 carbon atoms, alkylthio of 1 to 4 carbon atoms, alkylsulfinyl of 1 to 4 carbon atoms, alkylsulfonyl of 1 to 4 carbon atoms, cyano, trifluoromethyl, trichloromethyl, phenoxy or substituted phenoxy of the formula ##STR3## wherein each Z independently represents chloro, fluoro, bromo, nitro, cyano, alkoxy of 1 to 4 carbon atoms or alkylthio of 1 to 4 carbon atoms, with the proviso that when either n is 2 or 3, all X groups are sterically compatible with each other and all Z groups are sterically compatible with each other; Y represents oxygen or sulfur; each n can independently represent an integer of from 0 to 3, inclusive; R.sup.1 represents hydrogen, chloro, fluoro, bromo, alkyl of 1 to 4 carbon atoms, cycloalkyl of 3-6 carbon atoms, phenyl, phenylthio, alkoxy of 1 to 4 carbon atoms, alkylthio of 1 to 4 carbon atoms, alkylsulfinyl of 1 to 4 carbon atoms, alkylsulfonyl of 1 to 4 carbon atoms, thiocyanato, trifluoromethyl, trichloromethyl, amino, mono- or dialkylamino wherein each alkyl group independently contains from 1 to 4 carbon atoms; R.sup.2 represents methyl, ethyl, propyl or isobutyl and R.sup.3 represents methoxy, ethoxy, propoxy, ethyl, mono- or dialkylamino wherein each alkyl group independently contains from 1 to 4 carbon atoms, alkylthio of 1 to 4 carbon atoms or phenyl.
摘要翻译：制备符合下式的化合物：其中R表示与下式之一相对应的含氮杂环基，每个X独立地表示氯，氟，溴，硝基，1至4个碳原子的烷基，氨基，单 - 或二烷基氨基，其中每个烷基独立地含有1至4个碳原子，1至4个碳原子的烷氧基，1至4个碳原子的烷硫基，1至4个碳原子的烷基亚磺酰基 1至4个碳原子的烷基磺酰基，氰基，三氟甲基，三氯甲基，苯氧基或取代的苯氧基，其中每个Z独立地表示氯，氟，溴，硝基，氰基，1-4个碳原子的烷氧基或烷硫基具有1至4个碳原子，条件是当n为2或3时，所有X基彼此在空间上相容，并且所有Z基彼此在空间上相容; Y表示氧或硫; 每个n可以独立地表示0至3的整数，包括0和3; R 1表示氢，氯，氟，溴，1至4个碳原子的烷基，3-6个碳原子的环烷基，苯基，苯硫基，1至4个碳原子的烷氧基，1至4个碳原子的烷硫基，1至 4个碳原子，1至4个碳原子的烷基磺酰基，硫氰酸酯，三氟甲基，三氯甲基，氨基，一或二烷基氨基，其中每个烷基独立地含有1至4个碳原子; R 2表示甲基，乙基，丙基或异丁基，R 3表示甲氧基，乙氧基，丙氧基，乙基，单 - 或二烷基氨基，其中各烷基独立地含有1至4个碳原子，1至4个碳原子的烷硫基或苯基。

64. 发明授权

US4260767A 2-Pyridylhydrazides 失效
标题翻译： 2-吡啶基酰肼
公开(公告)号：US4260767A
公开(公告)日：1981-04-07
申请号：US106789
申请日：1979-12-26
申请人： John P. Dusza
发明人： John P. Dusza
IPC分类号： C07D213/77
CPC分类号： C07D213/77
摘要： 2-Pyridylhydrazides useful as antiinflammatory agents.
摘要翻译：用作抗炎剂的2-吡啶基酰肼。

65. 发明授权

US4254128A 2-Adamantyl hydrazines and biocidal compositions thereof 失效
标题翻译： 2-金刚烷基肼及其杀生物组合物
公开(公告)号：US4254128A
公开(公告)日：1981-03-03
申请号：US963113
申请日：1978-11-22
申请人： Ben-Zion Weiner , Raul Suchi , Jeffrey Sterling , Haim Yellin
发明人： Ben-Zion Weiner , Raul Suchi , Jeffrey Sterling , Haim Yellin
IPC分类号： A61K31/15 , A01N45/00 , A61K31/185 , A61K31/195 , A61K31/215 , A61K31/445 , A61P31/04 , A61P31/10 , A61P31/12 , C07C67/00 , C07C241/00 , C07C243/20 , C07C243/22 , C07D213/77 , C07D215/28 , C07D215/42 , C07D233/80 , C07D295/22 , C07D295/30 , C07D327/06 , A61K31/40
CPC分类号： C07D213/77 , C07C243/00 , C07D215/42 , C07D233/80 , C07D295/30
摘要： The invention provides novel 2-adamantyl hydrazine derivatives of the general formula A ##STR1## In this formula R.sub.1 is hydrogen or a lower alkyl group of 1-4 carbon atoms; R.sub.2 and R.sub.3 are the same or different and are each hydrogen, an unsubstituted or substituted radical being a lower alkyl of 1-4 carbon atoms, a lower alkanoic acid radical of 2-4 carbon atoms or a lower alkyl ester thereof, adamantyl, aryl, aralkyl, in which the alkyl moiety has from 1-4 carbon atoms or an unsubstituted or substituted heterocyclic radical of aromatic character; or R.sub.2 and R.sub.3 together with the nitrogen atom to which they are attached form an unsubstituted or substituted non-aromatic cyclic radical.The invention further provides pharmaceutically acceptable acid addition salts of the above compounds.Several methods of preparation of the new compounds are described.The novel compounds according to the invention possess valuable antifungal (human and plant), antiviral, antiprotozoal and antimicrobial properties.
摘要翻译：本发明提供了通式为A的新型2-金刚烷基肼衍生物。在该式中，R 1是氢或1-4个碳原子的低级烷基; R2和R3相同或不同，各自为氢，未取代或取代的基团为1-4个碳原子的低级烷基，2-4个碳原子的低级链烷酸基团或其低级烷基酯，金刚烷基，芳基，其中烷基部分具有1-4个碳原子的芳烷基或芳族特征的未取代或取代的杂环基; 或R 2和R 3与它们所连接的氮原子一起形成未取代或取代的非芳族环状基团。本发明进一步提供上述化合物的药学上可接受的酸加成盐。描述了几种制备新化合物的方法。根据本发明的新化合物具有有价值的抗真菌（人和植物），抗病毒，抗原虫和抗微生物特性。

66. 发明授权

US4242515A Substituted 3-alkyl-6-phenyl-1,2,4-triazolo-[4,3-a]pyridines 失效
标题翻译：取代的3-烷基-6-苯基-1,2,4-三唑并 - [4,3-a]吡啶
公开(公告)号：US4242515A
公开(公告)日：1980-12-30
申请号：US24849
申请日：1979-03-28
申请人： Ronald I. Trust , Jay D. Albright
发明人： Ronald I. Trust , Jay D. Albright
IPC分类号： G11C7/00 , A61K31/435 , A61P25/20 , C07D213/61 , C07D213/64 , C07D213/77 , C07D213/80 , C07D213/82 , C07D213/85 , C07D471/04 , G11C11/34 , G11C11/4063 , G11C11/4091 , A61K31/41
CPC分类号： C07D213/64 , C07D213/61 , C07D213/77 , C07D213/80 , C07D213/82 , C07D213/85 , C07D471/04 , G11C11/4063 , G11C11/4091
摘要： This disclosure describes novel 3-alkyl-6-(substituted-phenyl)-1,2,4-triazolo[4,3-a]pyridines useful as anxiolytic agents.
摘要翻译：本公开描述了可用作抗焦虑剂的新型3-烷基-6-（取代 - 苯基）-1,2,4-三唑并[4,3-a]吡啶。

67. 发明授权

US4209626A Substituted 6-phenyl-1,2,4-triazolo[4,3-a]pyridines 失效
标题翻译：取代的6-苯基-1,2,4-三唑并[4,3-a]吡啶
公开(公告)号：US4209626A
公开(公告)日：1980-06-24
申请号：US20886
申请日：1979-03-15
申请人： Ronald I. Trust , Jay D. Albright
发明人： Ronald I. Trust , Jay D. Albright
IPC分类号： C07D213/61 , C07D213/64 , C07D213/77 , C07D213/80 , C07D213/82 , C07D213/85 , C07D471/04 , A61K31/44
CPC分类号： C07D213/64 , C07D213/61 , C07D213/77 , C07D213/80 , C07D213/82 , C07D213/85 , C07D471/04
摘要： This disclosure describes novel 6-(substituted-phenyl)-1,2,4-triazolo[4,3-a]pyridines useful as hypotensive agents.
摘要翻译：本公开描述了用作低血压剂的新型6-（取代苯基）-1,2,4-三唑并[4,3-a]吡啶。

68. 发明授权

US4083984A 1-Substituted phenyl-4(1H)-pyridinone hydrazones and composition therewith for treatment of coccidiosis 失效
标题翻译： 1-取代的苯基-4（1H） - 吡啶酮腙及其组合物用于治疗球虫病
公开(公告)号：US4083984A
公开(公告)日：1978-04-11
申请号：US813930
申请日：1977-07-08
申请人： Michael H. Fisher , William V. Ruyle
发明人： Michael H. Fisher , William V. Ruyle
IPC分类号： C07D213/20 , C07D213/68 , C07D213/77 , A01N9/22 , C07D211/18
CPC分类号： C07D213/77 , C07D213/20 , C07D213/68
摘要： Novel 1-substitutedphenyl-4(1H)-pyridinone hydrazones are prepared by reacting 1-substitutedphenyl-4(1H)-pyridinone hydrazone with substituted benzaldehydes. The novel hydrazones are useful as anticoccidial agents.
摘要翻译：通过1-取代苯基-4（1H） - 吡啶酮腙与取代的苯甲醛反应来制备新的1-取代苯基-4（1H） - 吡啶酮腙。新颖的腙可用作抗球虫剂。

69. 发明授权

US3927003A 6-Hydrazino-2,3,5-trihalo-4-alkylthio pyridines 失效
标题翻译： 6-肼基-2,3,5-三卤代-4-烷硫基吡啶
公开(公告)号：US3927003A
公开(公告)日：1975-12-16
申请号：US53679074
申请日：1974-12-27
申请人： DOW CHEMICAL CO
发明人： RUETMAN SVEN H , WATSON RICHARD N
IPC分类号： C08K5/00 , A01N43/40 , C07D213/70 , C07D213/71 , C07D213/77 , C08K5/36
CPC分类号： C07D213/77 , C07D213/70 , C07D213/71
摘要： Novel compounds having the formula

WHEREIN R is an alkyl group of 1 to 5 carbons, X is Br or Cl and Y is Cl or is Br except when X is Cl, are prepared by the reaction of a hydrazine source material with a corresponding compound of the formula

The product compounds are fungicidal in their own right and are readily oxidized to highly active trihalo-4-alkylsulfonyl pyridine fungicides.
摘要翻译：具有式WHEREIN R的新型化合物是1至5个碳的烷基，X是Br或Cl，Y是Cl或是Br，除了当X是Cl时，是通过肼源材料与相应的化合物该化合物产物化合物本身是杀真菌剂，并且容易被氧化成高活性三卤代-4-烷基磺酰基吡啶类杀真菌剂。

70. 发明授权

US3818104A Use of dithiobiurets as fungicides 失效
标题翻译：二氢AS。。。。。。。
公开(公告)号：US3818104A
公开(公告)日：1974-06-18
申请号：US10036570
申请日：1970-12-21
申请人： EXXON RESEARCH ENGINEERING CO
发明人： ZIELINSKI J
IPC分类号： C07C335/40 , C07D209/08 , C07D209/48 , C07D209/76 , C07D213/40 , C07D213/77 , C07D231/08 , C07D307/14 , C07D307/52 , C07D521/00 , A01N9/12
CPC分类号： C07D213/77 , C07C335/40 , C07C2601/14 , C07D209/08 , C07D209/48 , C07D209/76 , C07D213/40 , C07D231/08 , C07D231/12 , C07D233/56 , C07D249/08 , C07D307/14 , C07D307/52
摘要： Semicarbazides, especially the tetraalkylated thiosemicarbazides, and biuret derivatives, especially the monoand di-thiobiuret derivatives, are effective fungicides, bactericides, herbicides, and also have demonstrated effective growth regulating activity. Exemplary of preferred semicarbazides are those of the general formula:

WHERE R1-R4 can be unsubstituted or substituted C1-C14 alkyl and X can be hydrogen, or unsubstituted or substituted C1-C14 alkyl and Y can be O or S. Exemplary of preferred biuret derivatives are those of the general formula:
WHEREIN R5-R11 can be hydrogen or unsubstituted or substituted C1-C14 alkyl and Y can be O or S and combinations thereof; and Q can be R9 or
摘要翻译：氨基脲，特别是四烷基化的氨基硫脲，和缩二脲衍生物，特别是单硫代硫代嘌呤衍生物和二硫代尿素衍生物，是有效的杀真菌剂，杀菌剂，除草剂，并且也已证明有效的生长调节活性。优选的氨基脲的实例是下列通式：

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