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82. 发明专利

JPS58128349A NOVEL N,N'-BIS-(BETA-HYDROXYALKYL)-ARYLAMINE DERIVATIVES 失效
公开(公告)号：JPS58128349A
公开(公告)日：1983-07-30
申请号：JP749383
申请日：1983-01-21
申请人： BAYER AG
发明人： EERITSUHI AIMERUSU , DEIITAA MARUGOTSUTE , RORUFU DAIN , KURAUSU KURAFUTO , BERUNAA KUREEKAA
IPC分类号： C08G73/00 , C07C67/00 , C07C213/00 , C07C217/32 , C07C219/04 , C07C219/12 , C08F299/04 , C08K5/18

83. 发明专利

JPS58118546A PREPARATION OF DICYCLOMINE HYDROCHLORIDE 失效
公开(公告)号：JPS58118546A
公开(公告)日：1983-07-14
申请号：JP100882
申请日：1982-01-08
申请人： KAWAKEN FINE CHEMICALS CO
发明人： KAGAWA HISASHI , KIMIZUKA YOSHIYUKI
IPC分类号： C07C219/12 , C07C51/00 , C07C61/13 , C07C67/00 , C07C213/00
摘要： PURPOSE:To prepare the titled compound in high yield, by reacting[1,1'-bicyclohexyl]-2-ol, etc. with formic acid, reacting the resultant carboxylic acid with 2-(diethylamino)ethyl chloride hydrochloride in the presence of a base, and converting the product to a salt. CONSTITUTION:[1,1'-Bicyclohexyl]-2-ol of formulaIand/or[1,1'-bicyclohexyl]-1-ol of formula II is made to react with formic acid in the presence of at least one kind of dehydrating agent selected from concentrated sulfuric acid, fuming sulfuric acid, phosphoric acid, and a mixture of phosphoric acid and phosphorus pentoxide to produce[1,1'-bicyclohexyl]-1-carboxylic acid of formula III. The reaction mixture is mixed with an aqueous solution of 2-(diethylamino)ethyl chloride hydrochloride, and an alkaline aqueous solution is added dropwise to the mixture to form the ester of formula IV, which is converted to the hydrochloride to obtain the compound of formula V.

84. 发明专利

JPS57122051A Preparation of(1,1'-bicyclohexyl)-1-carboxylic acid 2-(diethylamino)ethyl ester 失效
标题翻译：（1,1'-二苄基）-1-羧酸2-（二乙基氨基）乙酯的制备
公开(公告)号：JPS57122051A
公开(公告)日：1982-07-29
申请号：JP747481
申请日：1981-01-21
申请人： Kawaken Fine Chem Co Ltd
发明人： KAGAWA HISASHI , KIMIZUKA YOSHIYUKI
IPC分类号： C07C219/12 , C07C67/00 , C07C213/00
摘要： PURPOSE: To prepare the titled compound useful as a remedy for the spasmodic diseases of the stomach and the gallbladder, by reacting a bicyclohexanol compound with formic acid, and reacting the product with 2-(diethylamino)ethyl chloride hydrochloride.
CONSTITUTION: The objective compound of formula IV can be obtained by (1) reacting [1,1'-bicyclohexyl]-2-ol of formulaI and/or [1,1'-bicyclohexyl]-1-ol of formula II with formic acid in the presence of conc. sulfuric acid, (2) adding an aqueous alkaline solution to the resultant [1,1'-bicyclohexyl]-1-carboxylic acid of formula III to convert the carboxylic acid to an aqueous solution of the alkali metal salt, and (3) esterifying with an aqueous solution of 2-(diethylamino) ethyl chloride hydrochloride.
COPYRIGHT: (C)1982,JPO&Japio
摘要翻译：目的：通过使双环己醇化合物与甲酸反应，并使产物与2-（二乙基氨基）乙基氯盐酸盐反应，制备可用作胃和胆囊痉挛性疾病的药物的标题化合物。结构式：式Ⅳ的目标化合物可以通过以下方法获得：（1）使式Ⅰ的[1，1'-二环己基] -2-醇和/或式Ⅱ的[1,1'-二环己基] -1-醇与甲酸酸在浓缩物存在下硫酸，（2）向所得的式III的[1,1'-双环己基] -1-羧酸加入碱性水溶液以将羧酸转化为碱金属盐的水溶液，和（3）酯化与2-（二乙基氨基）乙基氯盐酸盐的水溶液。

85. 发明专利

JPS5788102A AGRICULTURAL FUNGICIDE 失效
公开(公告)号：JPS5788102A
公开(公告)日：1982-06-01
申请号：JP16341180
申请日：1980-11-21
申请人： MITSUI TOATSU CHEMICALS , HARIMA CHEMICALS INC
发明人： KOUSHI MASATO , FUJII RIYOUICHI , ISHIHARA KOUICHI , TACHIBANA HAJIME , SHIMOTORI HITOSHI
IPC分类号： C07D251/18 , A01N37/08 , A01N37/32 , A01N37/34 , A01N37/52 , A01N43/66 , A01N43/68 , A01N47/12 , A01N47/18 , A01N47/22 , C07C51/00 , C07C61/39 , C07C67/00 , C07C213/00 , C07C219/12 , C07C231/00 , C07C233/38 , C07C239/00 , C07C253/00 , C07C255/46 , C07C257/18 , C07C271/22 , C07D209/66 , C07D307/77
摘要： PURPOSE:An agricultural fungicide having an improved germicidal action and a propagation inhibiting action on various kinds of plant pathogenic germs, especially exhibiting excellent exterminating action on blast of rice plant, having low toxicity and no phytotoxicity, comprising one or more of specific abietic acid derivatives as active ingredients. CONSTITUTION:A fungicide comprising an abietic acid derivative, e.g., dehydroabiethylchloline iodide, N-phenyldehydroabiethylamidine, etc., comprising 5alpha, 10beta type A/B bonded ring, or 5alpha, 10beta type A/B bonded ring shown by the formula Ior formula II (R is H, OH, acryl, acyloxy, carbamyloxy; R is H or isopropyl; R is nitrile, carboxyl, methoxycarbonyl, carbamic ester, amide, triazyl, amidine, choline ester; R is carboxyl, methoxycarbonyl; R is O, imino, alkylamino, alkylaminoalkyl, phenyl, etc.).

86. 发明专利

JPS566414B2 失效
公开(公告)号：JPS566414B2
公开(公告)日：1981-02-10
申请号：JP14679276
申请日：1976-12-06
IPC分类号： A61K31/215 , A61K31/415 , A61K31/42 , A61K31/421 , A61K31/425 , A61K31/426 , A61K31/535 , A61K31/5377 , A61P9/00 , A61P9/06 , A61P25/24 , A61P25/26 , C07C67/00 , C07C69/74 , C07C213/00 , C07C219/12 , C07C219/34 , C07D233/02 , C07D233/06 , C07D239/04 , C07D263/04 , C07D263/12 , C07D265/08 , C07D277/04 , C07D277/10

87. 发明专利

JPS5377043A DERIVATIVE OF AZULENYL AMINOGLYOXYLATE 失效
公开(公告)号：JPS5377043A
公开(公告)日：1978-07-08
申请号：JP15220576
申请日：1976-12-17
申请人： ORIENTAL PHARM SYNTH CHEM
发明人： HAMASHIMA MAKOTO , OKUDA HIROHISA
IPC分类号： C07D295/08 , A61K31/215 , A61K31/40 , A61K31/44 , A61K31/4402 , A61K31/4406 , A61K31/4409 , A61K31/4418 , A61K31/445 , A61K31/535 , A61K31/5375 , A61P1/04 , C07C67/00 , C07C213/00 , C07C219/12 , C07D211/42 , C07D211/44 , C07D211/46 , C07D213/30 , C07D213/65 , C07D213/68 , C07D295/14

89. 发明专利

JPS504652B1 失效
公开(公告)号：JPS504652B1
公开(公告)日：1975-02-22
申请号：JP2723167
申请日：1967-04-28
IPC分类号： C07D295/08 , A61K31/215 , A61M5/178 , C07C62/04 , C07C219/12 , C07D211/08 , C07D211/42 , C07D211/90 , C07D295/10 , C07D295/14 , C07C93/197 , A61K31/445 , A61K31/495 , A61K31/535 , C07D211/36

90. 发明申请

WO2005005345A3 USE OF FUNCTIONALIZED ONIUM SALTS AS A SOLUBLE SUPPORT FOR ORGANIC SYNTHESIS 审中-公开
标题翻译：作为有机合成的可溶性支持使用功能性的盐水
公开(公告)号：WO2005005345A3
公开(公告)日：2005-03-31
申请号：PCT/FR2004001724
申请日：2004-07-02
申请人： CENTRE NAT RECH SCIENT , UNIV RENNES , VAULTIER MICHEL , GMOUH SAID , HASSINE FATIMA
发明人： VAULTIER MICHEL , GMOUH SAID , HASSINE FATIMA
IPC分类号： C07B37/02 , C07B37/04 , C07B37/12 , C07B61/00 , C07C67/03 , C07D211/16 , C07C209/08 , C07C211/63 , C07C213/02 , C07C213/08 , C07C215/44 , C07C219/10 , C07C219/12
CPC分类号： C07D211/16 , C07B37/02 , C07B37/04 , C07B37/12 , C07B61/00 , C07C67/03 , C07C2602/42 , C07C69/76 , C07C69/618 , C07C69/753 , C07C69/92
摘要： The invention relates to the use of a onium salt functionalized by at least one organic function, as a soluble support, in the presence of at least one organic solvent, for organic synthesis of a molecule, in a homogenous phase, by at least one transformation of said organic function. The onium salt enables the synthesized molecule to be released. The onium salt is present in liquid or solid form at room temperature and corresponds to formula Al , X1 , wherein A1 represents a cation and X1 représents an anion.
摘要翻译：本发明涉及在至少一种有机功能上作为可溶性载体在至少一种有机溶剂的存在下官能化的鎓盐的用途，用于通过至少一种转化在均相中有机合成分子的有机功能。鎓盐使得合成的分子被释放。鎓盐在室温下以液体或固体形式存在，对应于式A1 + X1，其中A1 +表示阳离子，X1'代表阴离子。

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