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31. 发明授权

US4761474A 3-(1H-tetrazol-5-yl)thieno[2,3-d]pyrimidin-4(3H)-ones 失效
标题翻译：（1H-四唑-5-基）噻吩并[2,3-d]嘧啶-4（3H） - 酮
公开(公告)号：US4761474A
公开(公告)日：1988-08-02
申请号：US833871
申请日：1986-02-25
申请人： Norton P. Peet , Shyam Sunder , Anna P. Vinogradoff
发明人： Norton P. Peet , Shyam Sunder , Anna P. Vinogradoff
IPC分类号： A61K31/505 , A61P11/00 , A61P27/16 , A61P37/08 , C07D333/00 , C07D409/12 , C07D495/02 , C07D495/04 , C07D513/04
CPC分类号： C07D495/04
摘要： 3-(1H-Tetrazol-5-yl)thieno[2,3-d]pyrimidin-4(3H)-ones useful as antiallergic agents are described herein. The compounds are prepared by cyclization of an appropriate substituted amidine using an alkali metal base. The reaction is carried out in an appropriate inert solvent.
摘要翻译：本文描述了可用作抗过敏剂的3-（1 H-四唑-5-基）噻吩并[2,3-d]嘧啶-4（3H）酮。通过使用碱金属碱使适当的取代的脒环化来制备化合物。该反应在合适的惰性溶剂中进行。

32. 发明申请

US20190152913A1 1,4-SUBSTITUTED PIPERIDINE DERIVATIVES 审中-公开
公开(公告)号：US20190152913A1
公开(公告)日：2019-05-23
申请号：US16257591
申请日：2019-01-25
申请人： 89BIO LTD
发明人： Nadine C. Becknell , Reddeppa Reddy Dandu , Bruce D. Dorsey , Dimitar B. Gotchev , Robert L. Hudkins , Linda Weinberg , Craig A. Zificsak , Allison L. Zulli
IPC分类号： C07D211/44 , C07D495/04 , C07D401/14 , C07D211/54 , C07D211/58 , C07D401/04 , C07D495/02 , C07D491/048 , C07D471/08 , C07D471/04 , C07D471/02 , C07D417/14 , C07D417/12 , C07D409/14 , C07D405/12 , C07D405/06 , C07D401/12 , C07D413/14 , C07D405/14 , C07D409/12
摘要： Described herein are 1,4-substituted piperidine compounds according to Formula I that have demonstrated activity as fatty acid synthase inhibitors. Also described herein are pharmaceutical compositions containing the described 1,4-substituted piperidine compounds, and methods of treating diseases mediated by fatty acid synthase, by administering one or more of the compounds or pharmaceutical formulations described herein. Also described herein are methods of synthesizing the compounds described, including the described 1,4-substituted piperidine compounds and synthetic intermediates useful in those syntheses.

33. 发明申请

US20190027701A1 ORGANIC TRANSISTOR AND GAS SENSOR 审中-公开
公开(公告)号：US20190027701A1
公开(公告)日：2019-01-24
申请号：US16077146
申请日：2017-06-01
申请人： LG CHEM, LTD.
发明人： Bogyu LIM , Yong-Young NOH , Jaechol LEE
IPC分类号： H01L51/05 , H01L51/00 , G01N27/414 , C07F7/08 , C07D487/02 , C07D495/02
摘要： The present specification relates to an organic transistor including an organic semiconductor layer including a compound, and a gas sensor to which the organic transistor is applied.

34. 发明授权

US09771355B2 Compositions and methods for the treatment of epilepsy and neurological disorders 有权
公开(公告)号：US09771355B2
公开(公告)日：2017-09-26
申请号：US14626931
申请日：2015-02-20
申请人： Mahesh Kandula
发明人： Mahesh Kandula
IPC分类号： A61K31/55 , C07D223/28 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D495/02
CPC分类号： C07D409/12 , C07D223/28
摘要： The invention relates to the compounds of formula I and formula Ia or its pharmaceutical acceptable polymorphs, solvates, enantiomers, stereoisomers and hydrates thereof. The pharmaceutical compositions comprising an effective amount of formula I or formula Ia; and methods for treating or preventing epilepsy, seizures and convulsions may be formulated for oral, buccal, rectal, topical, transdermal, transmucosal, intravenous, parenteral administration, syrup, or injection. Such compositions may be used to treatment of epilepsy, seizures and convulsions.

35. 发明授权

US09133210B2 Compounds and pharmaceutical compositions thereof for the treatment of cystic fibrosis 有权
标题翻译：用于治疗囊性纤维化的化合物及其药物组合物
公开(公告)号：US09133210B2
公开(公告)日：2015-09-15
申请号：US14451619
申请日：2014-08-05
申请人： Galapagos NV
发明人： Steven Emiel Van Der Plas , Hans Kelgtermans , Sébastien Jean Jacques Cédric Dropsit Montovert , Sébastien Laurent Xavier Martina , Martin James Inglis Andrews
IPC分类号： C07D495/02 , C07D495/04 , C07F9/6561 , A61K31/38
CPC分类号： A61K31/381 , A61K31/38 , A61K31/4025 , A61K31/4155 , A61K31/4162 , A61K31/4178 , A61K31/4196 , A61K31/422 , A61K31/427 , A61K31/436 , A61K31/437 , A61K31/4436 , A61K31/497 , A61K31/501 , A61K31/517 , A61K31/519 , A61K31/53 , A61K31/675 , C07D495/04 , C07F7/0812 , C07F9/091 , C07F9/6561
摘要： The present invention discloses compounds according to Formula I: wherein R1 is as defined herein. The present invention relates to compounds and their use in the treatment of cystic fibrosis, methods for their production, pharmaceutical compositions comprising the same, and methods of treatment cystic fibrosis by administering a compound of the invention.
摘要翻译：本发明公开了根据式I的化合物：其中R 1如本文所定义。本发明涉及化合物及其在治疗囊性纤维化中的用途，其制备方法，包含其的药物组合物和通过施用本发明化合物治疗囊性纤维化的方法。

36. 发明授权

US08941007B2 Electron donating polymer and organic solar cell including the same 有权
标题翻译：给电子聚合物和包括其的有机太阳能电池
公开(公告)号：US08941007B2
公开(公告)日：2015-01-27
申请号：US13421198
申请日：2012-03-15
申请人： Soo-Ghang Ihn , Yeong-Suk Choi , Youn-Hee Lim , Bulliard Xavier , Sung-Young Yun , In-Sun Park , Yeon-Ji Chung
发明人： Soo-Ghang Ihn , Yeong-Suk Choi , Youn-Hee Lim , Bulliard Xavier , Sung-Young Yun , In-Sun Park , Yeon-Ji Chung
IPC分类号： H01L31/00 , C08G63/688 , C07D333/00 , C07D495/02 , H01L51/00 , H01L51/42
CPC分类号： H01L51/0036 , B82Y10/00 , H01L51/0047 , H01L51/4253 , Y02E10/549
摘要： A polymer, and an organic solar cell including the polymer, include a repeating unit A represented by Chemical Formula 1, and a repeating unit B represented by Chemical Formula 2.
摘要翻译：聚合物和包含该聚合物的有机太阳能电池包括由化学式1表示的重复单元A和由化学式2表示的重复单元B.

37. 发明授权

US08710245B2 Multicyclic compounds and methods of use thereof 有权
标题翻译：多环化合物及其使用方法
公开(公告)号：US08710245B2
公开(公告)日：2014-04-29
申请号：US13513176
申请日：2010-12-03
申请人： Liming Shao , John Emmerson Campbell , Michael Charles Hewitt , Una Campbell , Taleen G. Hanania
发明人： Liming Shao , John Emmerson Campbell , Michael Charles Hewitt , Una Campbell , Taleen G. Hanania
IPC分类号： C07D495/02 , A61K31/38 , C07D495/04
CPC分类号： A61K31/381 , A61K31/435 , A61K31/55 , A61K45/06 , C07D277/60 , C07D333/54 , C07D333/76 , C07D333/78 , C07D495/04 , C07D495/20
摘要： Provided herein are multicyclic compounds, methods of their synthesis, pharmaceutical compositions comprising the compounds, and methods of their use. The compounds provided herein are useful for the treatment, prevention, and/or management of various neurological disorders, including but not limited to, psychosis and schizophrenia.
摘要翻译：本文提供多环化合物，其合成方法，包含该化合物的药物组合物及其使用方法。本文提供的化合物可用于治疗，预防和/或治疗各种神经障碍，包括但不限于精神病和精神分裂症。

38. 发明授权

US08680296B2 Leaving substituent-containing compound, products produced using the same, and methods for producing the products 有权
标题翻译：离开含取代基的化合物，使用其制备的产物，以及制备该产品的方法
公开(公告)号：US08680296B2
公开(公告)日：2014-03-25
申请号：US13391448
申请日：2010-09-09
申请人： Daisuke Goto , Satoshi Yamamoto , Toshiya Sagisaka , Takuji Kato , Takashi Okada , Masato Shinoda , Shinji Matsumoto , Masataka Mohri , Keiichiro Yutani
发明人： Daisuke Goto , Satoshi Yamamoto , Toshiya Sagisaka , Takuji Kato , Takashi Okada , Masato Shinoda , Shinji Matsumoto , Masataka Mohri , Keiichiro Yutani
IPC分类号： C07D495/02 , H01J1/62
CPC分类号： H01L51/0052 , C07C1/213 , C07C15/20 , C07C15/24 , C07C15/28 , C07C15/38 , C07C15/56 , C07C15/58 , C07C15/60 , C07C17/093 , C07C17/10 , C07C17/361 , C07C25/22 , C07C69/013 , C07C69/18 , C07C69/63 , C07C2602/10 , C07C2603/24 , C07C2603/44 , C07C2603/50 , C07C2603/52 , C07D321/00 , C07D409/14 , C07D495/04 , C07D495/06 , H01L51/0074 , H01L51/0558
摘要： A leaving substituent-containing compound including a partial structure represented by the following General Formula (I): where a pair of X1 and X2 or a pair of Y1 and Y2 each represent a hydrogen atom; the other pair each represent a group selected from the group consisting of a halogen atom and a substituted or unsubstituted acyloxy group having one or more carbon atoms; a pair of the acyloxy groups represented by the pair of X1 and X2 or the pair of Y1 and Y2 may be identical or different, or may be bonded together to form a ring; R1 to R4 each represent a hydrogen atom or a substituent; and Q1 and Q2 each represent a hydrogen atom, a halogen atom or a monovalent organic group, and may be bonded together to form a ring.
摘要翻译：含有由以下通式（I）表示的部分结构的含有取代基的化合物：其中一对X1和X2或一对Y1和Y2各自表示氢原子; 另一对各自表示选自卤原子和具有一个或多个碳原子的取代或未取代的酰氧基的基团; 由一对X1和X2表示的一对酰氧基或一对Y1和Y2可以相同或不同，或者可以结合在一起形成环; R 1〜R 4各自表示氢原子或取代基; 并且Q1和Q2各自表示氢原子，卤素原子或一价有机基团，并且可以结合在一起形成环。

39. 发明授权

US08273269B2 Red colour filter composition 有权
标题翻译：红色滤色片组成
公开(公告)号：US08273269B2
公开(公告)日：2012-09-25
申请号：US12993095
申请日：2009-05-05
申请人： Roman Lenz , Gerardus De Keyzer , Mathias Duggeli , Patrick Christopher Holzhuter
发明人： Roman Lenz , Gerardus De Keyzer , Mathias Duggeli , Patrick Christopher Holzhuter
IPC分类号： G02B5/23 , C07D487/02 , C07D491/02 , C07D495/02 , C07D497/02
CPC分类号： C09B57/004 , C09B67/0033 , C09B67/0039 , C09B69/00 , G02B5/223
摘要： A composition, for producing dispersions, thermoplastic masses and/or color filters, comprising (a) a colorant of formula (1) wherein 20-100 mol % R1 are Br and 80-100 mol % R3 are H, especially of formula (Ib) and/or (Ic); (b) from 0 to 150% by weight, based on (a), of C. I. Pigment Red 144, 188, 190, 224, 242 or 2,4,6-trimethylphenylperylene diimide; (c) from 3 to 25% by weight, based on (a), of a di- or tri-azacyclopentylmethyl-substituted colorant (formulae given); (d) from 0 to 10% by weight, preferably from 0.01 to 8% by weight, based on the sum of (a) and (b), of an additionally sulfonated colorant of the same kernels as in (c); and (e) from 0 to 30% by weight, preferably from 3 to 25% by weight, especially from 5 to 20% by weight, based on (a), of a diketopyrrolopyrrole colorant substituted by at least one chain containing a plurality of nitrogen atoms (cf. formula (V)).
摘要翻译：一种用于生产分散体，热塑性物质和/或滤色剂的组合物，其包含（a）式（1）的着色剂，其中20-100摩尔％的R 1是Br，80-100摩尔％的R 3是H，特别是式）和/或（Ic）; （b）基于（a）0-150重量％的C.I.颜料红144,188,190,224,242或2,4,6-三甲基苯基亚苯基二酰亚胺; （c）基于（a）3至25重量％的二 - 或三 - 氮杂环戊基甲基取代的着色剂（给出公式）; （d）相对于（c）中相同核的另外的磺化着色剂，基于（a）和（b）的总和为0至10重量％，优选为0.01至8重量％和（e）基于（a）0至30重量％，优选3至25重量％，特别是5至20重量％的由至少一个链取代的二酮吡咯并吡咯着色剂，所述链含有多个氮原子（参见式（Ⅴ））。

40. 发明授权

US08232546B2 Fused polycyclic aromatic compound, process for producing the same, and use thereof 有权
标题翻译：稠合多环芳香族化合物，其制造方法及其用途
公开(公告)号：US08232546B2
公开(公告)日：2012-07-31
申请号：US12312083
申请日：2007-10-22
申请人： Kazuo Takimiya , Tatsuya Yamamoto
发明人： Kazuo Takimiya , Tatsuya Yamamoto
IPC分类号： H01L51/00 , C07D495/02 , C07D517/02
CPC分类号： H01L51/0071 , C07C319/14 , C07C319/20 , C07C391/02 , C07D495/04 , C07D517/04 , H01L51/0074 , H01L51/0558 , Y10S428/917 , C07C321/28 , C07C323/22
摘要： In one embodiment of the present invention, a novel fused polycyclic aromatic compound of the present invention is (a) a compound including a benzodichalcogenophenobenzodichalcogenophene (BXBX) skeleton further having an aromatic ring(s) located outside the BXBX skeleton, or (b) a compound including a BXBX skeleton in which a benzene ring is substituted with a heterocyclic ring. The compound can strengthen intermolecular interaction due to greater π electron orbits. This improves an electron field effect mobility of an organic semiconductor device that is manufactured by use of the compound as an organic semiconductor material. Further, since the number of fused rings included in the compound is small, the compound does not cause problems that generally occur in compounds having an extremely large number of fused rings, i.e., poor solubility in solvent and poor atmospheric stability due to high affinity to oxygen. As a result, the fused polycyclic aromatic compound of the present invention can be preferably used as an organic semiconductor material.
摘要翻译：在本发明的一个实施方案中，本发明的新型稠合多环芳香族化合物是（a）还含有位于BXBX骨架外侧的芳香环的苯并二硫代苯并苯并二硫代苯并（BXBX）骨架的化合物，或（b）包括其中苯环被杂环取代的BXBX骨架的化合物。该化合物可以增强分子间的相互作用，电子轨道。这提高了通过使用化合物作为有机半导体材料制造的有机半导体器件的电子场效应迁移率。此外，由于化合物中包含的稠合环的数量少，所以化合物不会产生通常发生在具有极大数目的稠环的化合物中的问题，即在溶剂中的溶解性差和由于高亲和力而导致的差的大气稳定性氧。结果，本发明的稠合多环芳族化合物可以优选用作有机半导体材料。

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