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81. 发明授权

US06965032B2 Substituted dihydro 3-halo-1h-pyrazole-5-carboxylates and their preparation and use 有权
标题翻译：取代的二氢-3-卤代-1H-吡唑-5-羧酸酯及其制备和用途
公开(公告)号：US06965032B2
公开(公告)日：2005-11-15
申请号：US10482458
申请日：2002-08-13
申请人： John Herbert Freudenberger
发明人： John Herbert Freudenberger
IPC分类号： A01N43/56 , A61K31/415 , A61K31/4439 , C07C251/76 , C07D213/77 , C07D231/06 , C07D231/08 , C07D231/12 , C07D231/14 , C07D231/16 , C07D231/22 , C07D401/04 , C07D403/04 , C07D413/04 , C07D413/14
CPC分类号： A01N43/56 , C07C251/76 , C07D213/77 , C07D231/06 , C07D231/08 , C07D231/14 , C07D231/16 , C07D401/04 , C07D413/04 , C07D413/14
摘要： This invention relates to a compound of Formula I, a method for its preparation and its use in the preparation of a compound of Formula II wherein R1, R2, R3, X and n are as defined in the disclosure. This invention also discloses preparation of compounds of Formula III wherein R1, R2, R6, R7, R8 and n are as defined in the disclosure. Also disclosed are certain intermediates of Formula 4 for the preparation of compounds of Formula I wherein X is N and R2, R3 and n are as defined in the disclosure.
摘要翻译：本发明涉及式I化合物，其制备方法及其在制备式II化合物中的用途，其中R 1，R 2，R 2， N 3，X和n如本公开中所定义。本发明还公开了式III化合物的制备，其中R 1，R 2，R 6，R 7， R 8和n如本公开所定义。还公开了用于制备式I化合物的式4的某些中间体，其中X是N且R 2，R 3和n如本公开所定义。

82. 发明申请

US20050203149A1 Insecticide containing hydrazone derivatives as the active ingredient and novel hydrazone derivates 失效
标题翻译：含腙衍生物作为活性成分的杀虫剂和新型腙衍生物
公开(公告)号：US20050203149A1
公开(公告)日：2005-09-15
申请号：US10500925
申请日：2003-01-10
申请人： Shinji Kawata , Shuko Okui , Shigeru Suzuki , Toshiki Fukuchi , Akiyuki Suwa
发明人： Shinji Kawata , Shuko Okui , Shigeru Suzuki , Toshiki Fukuchi , Akiyuki Suwa
IPC分类号： C07D237/12 , A01N37/18 , A01N37/50 , A01N43/08 , A01N43/10 , A01N43/40 , A01N43/54 , A01N43/58 , A01N43/60 , A01N43/78 , A01N43/80 , C07C251/76 , C07C255/66 , C07C257/02 , C07C323/41 , C07C323/48 , C07D213/40 , C07D213/61 , C07D213/68 , C07D213/74 , C07D213/75 , C07D213/77 , C07D239/30 , C07D241/12 , C07D261/10 , C07D277/20 , C07D277/30 , C07D277/32 , C07D277/82 , C07D307/16 , C07D307/52 , C07D333/24 , C07D333/28 , C07D417/12 , A01N37/34 , A01N43/36
CPC分类号： C07D213/40 , A01N37/50 , A01N43/08 , A01N43/10 , A01N43/40 , A01N43/54 , A01N43/58 , A01N43/60 , A01N43/78 , A01N43/80 , C07C251/76 , C07D213/61 , C07D213/68 , C07D213/74 , C07D213/75 , C07D213/77
摘要： A insecticide characterized by containing as active ingredient a hydrazone derivative of formula (I) wherein A and Q are an aryl or a heterocyclic group, W is oxygen atom, an aminylene, an alkylene group, an oxyalkylene group or an alkyleneoxy, X1 and X2 are hydrogen atom, an alkyl, an alkenyl, an alkynyl, an aryl, a heterocyclic group, formyl, an acyl, an alkoxycarbonyl, an aryloxycarbonyl, a heterocyclic oxycarbonyl, an alkylsulfinyl, an arylsulfinyl, a heterocyclic sulfinyl, an alkylsulfonyl, an arylsulfonyl or a heterocyclic sulfonyl, Y is oxygen atom or sulfur atom, Z is hydrogen atom, a halogen atom, cyano, an alkyl, an alkenyl, an alkynyl, an amino, an alkoxy or an alkylthio, the substituents may be substituted; and novel hydrazon derivatives.
摘要翻译：一种杀虫剂，其特征在于含有作为活性成分的式（I）腙衍生物，其中A和Q为芳基或杂环基，W为氧原子，亚氨基，亚烷基，氧化烯基或亚烷基氧基，X ^{1和X 2是氢原子，烷基，烯基，炔基，芳基，杂环基，甲酰基，酰基，烷氧基羰基，芳氧基羰基，杂环氧基羰基，烷基亚磺酰基，芳基亚磺酰基，杂环亚磺酰基，烷基磺酰基，芳基磺酰基或杂环磺酰基，Y是氧原子或硫原子，Z是氢原子，卤素原子，氰基，烷基，烯基，炔基，氨基，烷氧基或烷硫基，取代基可以被取代; 和腙衍生物。}

83. 发明申请

US20050165062A1 Substituted polycyclic aryl and heteroaryl pyridones useful for selective inhibition of the coagulation cascade 审中-公开
标题翻译：用于选择性抑制凝血级联的取代的多环芳基和杂芳基吡啶酮
公开(公告)号：US20050165062A1
公开(公告)日：2005-07-28
申请号：US11009787
申请日：2004-12-10
申请人： Michael South , Qingping Zeng , Ashton Hamme , Melvin Rueppel
发明人： Michael South , Qingping Zeng , Ashton Hamme , Melvin Rueppel
IPC分类号： C07D213/74 , C07D213/75 , C07D213/77 , C07D215/38 , C07D401/12 , C07D417/12 , C07D521/00 , A61K31/4439 , A61K31/4415 , C07D211/84 , C07D41/02
CPC分类号： C07D213/74 , C07D213/75 , C07D213/77 , C07D215/38 , C07D231/12 , C07D233/56 , C07D249/08 , C07D401/12 , C07D417/12
摘要： The invention relates to substituted polycyclic aryl and heteroaryl pyridone compounds useful as inhibitors of serine proteases of the coagulation cascade and compounds, compositions and methods for anticoagulant therapy for the treatment and prevention of a variety of thrombotic conditions including coronary artery and cerebrovascular diseases.
摘要翻译：本发明涉及用作凝血级联丝氨酸蛋白酶抑制剂的取代多环芳基和杂芳基吡啶酮化合物，以及用于治疗和预防各种血栓形成病症（包括冠状动脉和脑血管疾病）的抗凝血治疗的化合物，组合物和方法。

84. 发明申请

US20050075372A1 Method for controlling particular insect pest by applying anthranilamide compounds 审中-公开
标题翻译：通过施用邻氨基苯甲酰胺化合物控制特定害虫的方法
公开(公告)号：US20050075372A1
公开(公告)日：2005-04-07
申请号：US10483115
申请日：2002-08-13
申请人： George Lahm , Stephen McCan , Kanu Patel , Thomas Selby , Thomas Stevenson
发明人： George Lahm , Stephen McCan , Kanu Patel , Thomas Selby , Thomas Stevenson
IPC分类号： A01N43/56 , A01N43/60 , A01N43/76 , A01N43/78 , A01N43/80 , A01N43/90 , A01N47/12 , A01N53/06 , A01N57/28 , A01N63/00 , A01P7/02 , C07C251/76 , C07D213/77 , C07D231/06 , C07D231/08 , C07D231/14 , C07D231/16 , C07D233/96 , C07D401/04 , C07D413/04 , C07D413/14 , A01N43/40
CPC分类号： A01N43/56 , A01N43/54 , A01N43/58 , A01N43/86 , C07C251/76 , C07D213/77 , C07D231/06 , C07D231/08 , C07D231/14 , C07D231/16 , C07D401/04 , C07D413/04 , C07D413/14
摘要： This invention pertains to a method for controlling lepidopteran, homopteran, hemipteran, thysanopteran and coleopteran insect pests comprising contacting the insects or their environment with an arthropodicidally effective amount of a compound of Formula I, its N-oxide or an agriculturally suitable salt thereof wherein A and B and R1 through R8 are as defined in the disclosure. This invention further relates to a bezoxazinone compound of Formula 10 wherein R4 through R8 are as defined in the disclosure, useful for preparation of a compound of Formula I.
摘要翻译：本发明涉及一种控制鳞翅目，同翅目，半翅目，鳞翅目和鞘翅目昆虫害虫的方法，包括使昆虫或其环境与节肢动物学有效量的式I化合物，其N-氧化物或农业上合适的盐接触，其中A 并且B和R 1至R 8如本公开所定义。本发明还涉及式10的唑嗪酮化合物，其中R 4至R 8如本公开所定义，可用于制备式I化合物。

85. 发明申请

US20040198984A1 Arthropodicidal anthranilamides 有权
标题翻译：节肢动物杀虫剂邻氨基苯甲酰胺
公开(公告)号：US20040198984A1
公开(公告)日：2004-10-07
申请号：US10483168
申请日：2004-01-07
发明人： George Philip Lahm , Thomas Paul Selby , Thomas Martin Stevenson
IPC分类号： C07D43/04
CPC分类号： A01N43/56 , A01N37/38 , A01N43/16 , A01N43/707 , C07C251/76 , C07D213/77 , C07D231/06 , C07D231/08 , C07D231/14 , C07D231/16 , C07D401/04 , C07D413/04 , C07D413/14
摘要： This invention provides compounds of Formula 1, their N-oxides and agriculturally suitable salts 1 wherein R1, R2, R3, R4a, R4b and R5 are as defined in the disclosure. Also disclosed are methods for controlling invertebrate pests comprising contacting the invertebrate pests or their environment with a biologically effective amount of a compound of Formula 1 or a composition comprising a compound of Formula 1.
摘要翻译：本发明提供式1化合物，其N-氧化物和农业上合适的盐，其中R 1，R 2，R 3，R 4a，R 4b和R 5如披露。还公开了用于控制无脊椎动物害虫的方法，包括使无脊椎害虫或其环境与生物有效量的式1化合物或包含式1化合物的组合物接触。

86. 发明授权

US06710180B2 Diazonium salts which are intermediates for 3-substituted pyridines 失效
标题翻译：作为3-取代吡啶的中间体的重氮盐
公开(公告)号：US06710180B2
公开(公告)日：2004-03-23
申请号：US10320591
申请日：2002-12-16
申请人： Dean Kent Hoglen
发明人： Dean Kent Hoglen
IPC分类号： C07D21376
CPC分类号： C07D213/77 , C07D213/63
摘要： The present invention relates to 3-substituted and 2,3-disubstituted pyridine compounds which are useful as intermediates in the synthesis of pyridylsulfonylurea herbicides. The invention also relates to arylation of alcohols using a pyridinediazonium salt. More particularly the arylation process of the instant invention relates to the synthesis of 2,3-disubstituted pyridine compounds via anhydrous diazotization of 3-amninopyridines to form a diazonium salt intermediate that is then reacted with the appropriate alcohol to produce the desired product. The invention additionally relates to pyridine-3-diazonium salt intermediates.
摘要翻译：本发明涉及可用作合成吡啶基磺酰脲除草剂的中间体的3-取代的和2,3-二取代的吡啶化合物。本发明还涉及使用吡啶并重氮盐的醇的芳基化。更具体地，本发明的芳基化方法涉及通过3-氨基吡啶的无水重氮化合成2,3-二取代的吡啶化合物以形成重氮盐中间体，然后与适当的醇反应以产生所需产物。本发明还涉及吡啶-3-重氮盐中间体。

87. 发明授权

US06645594B1 Formazan metal complex 失效
标题翻译：甲an金属络合物
公开(公告)号：US06645594B1
公开(公告)日：2003-11-11
申请号：US09762535
申请日：2001-02-08
申请人： Kentaro Yano , Katsumi Orita , Toshio Kawata , Shigeo Yasui
发明人： Kentaro Yano , Katsumi Orita , Toshio Kawata , Shigeo Yasui
IPC分类号： B32B302
CPC分类号： C07D213/77 , C07D213/86 , C07D213/87 , C07D401/14 , C07D405/12 , C07D417/14 , C09B50/00 , C09B50/04 , C09B67/0033 , G11B7/244 , G11B7/249 , Y10T428/21
摘要： The present invention provides organic compounds which improve the light resistance of organic dye compounds without substantially deteriorating their preferable light properties when applied to them, and have satisfactory solubility in organic solvents and compatibility with organic dye compounds. The object of the present invention is solved by formazan metal compounds which comprise specific formazan compounds as ligands; process thereof; light-resistant improvers, optical recording media, and light absorbents, which all comprise the formazan metal complexes; and formazan compounds as intermediates for producing the formazan metal complexes
摘要翻译：本发明提供了有机化合物，当施加到有机染料化合物上时，其有机染料化合物的耐光性能基本上不会劣化，而且在有机溶剂中的溶解性良好，与有机染料化合物的相容性提高。本发明的目的是通过包含特异性甲an化合物作为配体的甲an金属化合物来解决; 其过程; 耐光改进剂，光学记录介质和光吸收剂，其均包含甲an金属络合物; 和甲an化合物作为生产甲an金属络合物的中间体

88. 发明申请

US20030124053A1 Radiopharmaceuticals for imaging infection and inflammation 审中-公开
公开(公告)号：US20030124053A1
公开(公告)日：2003-07-03
申请号：US10151663
申请日：2002-05-20
发明人： John Andrew Barrett , Edward Hollister Cheesman , Thomas David Harris , Shuang Liu , Milind Rajopadhye , Michael Sworin
IPC分类号： A61K051/00 , C07D43/02
CPC分类号： C07F9/65583 , A61K51/0455 , A61K51/0478 , A61K51/0497 , C07C59/90 , C07C323/41 , C07D213/64 , C07D213/71 , C07D213/77 , C07D213/82 , C07D401/06 , C07D401/12 , C07D401/14 , C07D405/04 , C07D405/12 , C07D405/14 , C07F13/005
摘要： The present invention provides novel radiopharmaceuticals useful for the diagnosis of infection and inflammation, reagents and kits useful for preparing the radiopharmaceuticals, methods of imaging sites of infection and/or inflammation in a patient, and methods of diagnosing diseases associated with infection or inflammation in patients in need of such diagnosis. The radiopharmaceuticals bind in vivo to the leukotriene B4 (LTB4) receptor on the surface of leukocytes which accumulate at the site of infection and inflammation. The reagents provided by this invention are also useful for the treatment of diseases associated with infection and inflammation.

89. 发明申请

US20030092914A1 PROCESS FOR PREPARING ALKANESULFONYL PYRIDINES 失效
标题翻译：制备烷酰基吡啶的方法
公开(公告)号：US20030092914A1
公开(公告)日：2003-05-15
申请号：US10259155
申请日：2002-09-27
发明人： Jolanta Nowakowski , Dieter Haag
IPC分类号： C07D213/62 , C07D213/72
CPC分类号： C07D401/04 , C07D213/71 , C07D213/77
摘要： A process for preparing alkanesulfonyl pyridines of the formula 1: 1 is disclosed, wherein R1 is as defined herein. The compounds of formula 1 are useful in the preparation of pyridyl-substituted pyrazoles used in the treatment and alleviation of inflammation and other inflammation associated disorders.
摘要翻译：公开了制备式1的烷磺酰基吡啶的方法：其中R 1如本文所定义。式1的化合物可用于制备用于治疗和缓解炎症和其它炎症相关疾病的吡啶基取代的吡唑

90. 发明申请

US20030092744A1 Novel compounds for the management of aging-related and diabetic vascular complications, process for their preparation and therapeutic uses thereof 失效
标题翻译：用于治疗老化相关和糖尿病血管并发症的新型化合物，其制备方法及其治疗用途
公开(公告)号：US20030092744A1
公开(公告)日：2003-05-15
申请号：US10214704
申请日：2002-08-09
申请人： TORRENT PHARMACEUTICALS LTD.
发明人： Alangudi Sankaranarayanan
IPC分类号： A61K031/44 , C07D213/56
CPC分类号： C07D213/77 , A61K31/4425 , A61K31/4436 , A61K31/444 , A61K45/06 , C07D213/82 , C07D213/87 , C07D409/14 , A61K2300/00
摘要： The invention discloses novel compounds of the pyridinium series useful for the management of diabetes and aging-related vascular complications, including kidney disease, nerve damage, atherosclerosis, retinopathy, dermatological disorders and discoloration of teeth, by breaking preformed AGE, of the general formula I, or pharmaceutically acceptable salts thereof, 1 wherein, R1, R2, R3, X and m are as defined in the specification. The invention also discloses, method for preparation of the novel compounds of the series and pharmaceutical composition having one or more compounds as defined above as active ingredients. The invention further discloses a method of treatment of a diabetic patient by administering the compounds as defined above, either singly or in combination with drugs for antidiabetic therapy.
摘要翻译：本发明公开了用于治疗糖尿病和衰老相关血管并发症的新颖化合物，其包括肾脏疾病，神经损伤，动脉粥样硬化，视网膜病变，皮肤病学和牙齿变色，通过破坏预先形成的AGE，通式I 或其药学上可接受的盐，其中R1，R2，R3，X和m如说明书中所定义。本发明还公开了制备该系列新化合物的方法和具有一种或多种如上所定义的化合物作为活性成分的药物组合物。本发明还公开了一种通过单独给药上述化合物或与用于抗糖尿病治疗的药物组合来治疗糖尿病患者的方法。

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