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1. 发明授权

US06312698B1 Anti-fungal formulation active against a broad spectrum of dermatophytoses 有权
标题翻译：抗真菌制剂对广泛的皮肤病菌具有活性
公开(公告)号：US06312698B1
公开(公告)日：2001-11-06
申请号：US09537148
申请日：2000-03-29
申请人： Sushil Kumar Shahi , Amritesh Chandra Shukla , Anupam Dikshit , Ashok Kumar Bajaj , Anil Kumar Singh , Sushil Kumar
发明人： Sushil Kumar Shahi , Amritesh Chandra Shukla , Anupam Dikshit , Ashok Kumar Bajaj , Anil Kumar Singh , Sushil Kumar
IPC分类号： A61K3578
CPC分类号： A61K36/53
摘要： The invention provides a novel anti-fungal formulation active against a broad spectrum of dermatophytoses, said formulation comprising at least about 1% by weight of oil extracted from Rabdosia melissoides and one or more vegetable oils, solvents and additives.
摘要翻译：本发明提供了一种针对广谱皮肤真菌病的活性物质的新型抗真菌制剂，所述制剂包含至少约1重量％的从马来酸甜菜碱提取的油和一种或多种植物油，溶剂和添加剂。

2. 发明授权

US09260781B2 Process to deposit diamond like carbon as surface of a shaped object 有权
标题翻译：沉积类似碳的钻石作为成形物体的表面的工艺
公开(公告)号：US09260781B2
公开(公告)日：2016-02-16
申请号：US13201210
申请日：2010-01-27
申请人： Sushil Kumar , Prakash Narain Dixit , Chandra Mohan Singh Rauthan
发明人： Sushil Kumar , Prakash Narain Dixit , Chandra Mohan Singh Rauthan
IPC分类号： C23C16/27 , C23C16/26 , B65D23/02 , C23C16/02 , C23C16/04 , C23C16/455 , C23C16/509 , H01J37/32
CPC分类号： C23C16/26 , B65D23/02 , C23C16/0272 , C23C16/045 , C23C16/45578 , C23C16/509 , H01J37/32091
摘要： A plasma based deposition process to deposit thin film on the inner surfaces of the shaped objects such as plastic or metallic object like bottles, hollow tubes etc. at room temperature has been developed. In present invention uniform hydrogenated amorphous carbon (also called Diamond-Like Carbon, DLC) films on inner surfaces of plastic bottles is successfully deposited. Applications of such product include entire food and drug industries. There is a huge demand of polyethylene terephthalate (PET) or polyethylene naphthalate (PEN)) bottles, meant for the storage of potable water, carbonated soft drinks, wines, medicines etc. However, the higher cost prohibits their wide, spread use. The cheaper alternative is to use plastic bottles inside coated with chemically inert material such as Diamond-Like Carbon (DLC) will be commercially viable. Inventor process can be scaled up for mass production. This process can also be used for coating on inner surface of metallic cane or tube with a carbide forming interlayer (like hydrogenated amorphous silicon) to get the DLC films with better adhesion to inner surface of metals.
摘要翻译：已经开发了在室温下在诸如塑料或金属物体（如瓶子，中空管等）的成形物体的内表面上沉积薄膜的等离子体沉积工艺。在本发明中，成功地沉积了塑料瓶内表面上均匀的氢化无定形碳（也称为金刚石碳，DLC）膜。这些产品的应用包括整个食品和药品行业。聚对苯二甲酸乙二醇酯（PET）或聚萘二甲酸乙二醇酯（PEN））瓶子的需求很大，用于储存饮用水，碳酸软饮料，葡萄酒，药品等。但是，更高的成本禁止其广泛使用。更便宜的替代方法是使用塑料瓶内涂覆有化学惰性材料，如金刚石碳（DLC），这在商业上是可行的。发明人流程可以扩大批量生产。该方法也可用于在金属手杖或管的内表面上涂覆碳化物形成中间层（如氢化非晶硅），以使DLC膜具有更好的金属内表面附着力。

3. 发明申请

US20140128613A1 A PROCESS FOR PREPARATION OF INTERMEDIATES OF DONEPEZIL HYDROCHLORIDE 审中-公开
标题翻译：一种制备二苯甲基氯化物中间体的方法
公开(公告)号：US20140128613A1
公开(公告)日：2014-05-08
申请号：US14006160
申请日：2012-03-22
申请人： Renugadevi Gurusamy , Mita Roy , Ramasubramanian Shanmuganathan , Ashutosh Jagtap , Sivaramakrishnan Hariharan , Sushil Kumar Mishra , Karuna Wankhede
发明人： Renugadevi Gurusamy , Mita Roy , Ramasubramanian Shanmuganathan , Ashutosh Jagtap , Sivaramakrishnan Hariharan , Sushil Kumar Mishra , Karuna Wankhede
IPC分类号： C07D213/50
CPC分类号： C07D213/50
摘要： The present invention provides a process for the preparation of key intermediate for the synthesis 5,6-dimethoxy-2-[[1-(phenylmethyl)-4-piperidinyl]methyl]-1-indanone hydrochloride (donepezil hydrochloride). The present invention particularly provides a process for the preparation of 5,6-dimethoxy-2-(4-pyridylmethylene)-1-indanone comprising condensation of 5,6-dimethoxy-1-indanone with 4-pyridinecarboxaldehyde using an alkali metal hydroxide as a mild base in the presence of demineralized water as a solvent at a temperature in the range of 15° C. to 45° C. to yield 5,6-dimethoxy-2-(4-pyridylmethylene)-1-indanone, which is subsequently benzylated using benzyl bromide in the presence of solvent at a reflux temperature to yield 1-benzyl-4-[(5,6-dimethoxy-1-indanone-2-yl)methylene]pyridinium bromide.
摘要翻译：本发明提供了制备合成5,6-二甲氧基-2 - [[1-（苯基甲基）-4-哌啶基]甲基] - 茚满酮盐酸盐（盐酸多奈哌齐）的关键中间体的方法。本发明特别提供一种制备5,6-二甲氧基-2-（4-吡啶基亚甲基）-1-二氢茚酮的方法，该方法包括使用碱金属氢氧化物将5,6-二甲氧基-1-二氢茚酮与4-吡啶甲醛缩合在15℃至45℃的温度下，作为溶剂的软化水存在下的温和碱，得到5,6-二甲氧基-2-（4-吡啶基亚甲基）-1-二氢化茚，其为随后使用苄基溴在溶剂存在下在回流温度下苄化，得到1-苄基-4 - [（5,6-二甲氧基-1-茚满酮-2-基）亚甲基]吡啶鎓溴化物。

4. 发明申请

US20140077854A1 SEQUENTIAL STATE ELEMENTS RADIATION HARDENED BY DESIGN 有权
标题翻译：按设计硬化的序列状态元素辐射
公开(公告)号：US20140077854A1
公开(公告)日：2014-03-20
申请号：US14031585
申请日：2013-09-19
申请人： Lawrence T. Clark , Sandeep Shambhulingaiah , Sushil Kumar , Chandarasekaran Ramamurthy
发明人： Lawrence T. Clark , Sandeep Shambhulingaiah , Sushil Kumar , Chandarasekaran Ramamurthy
IPC分类号： H03K3/356 , G06F17/50
CPC分类号： H03K3/356086 , G06F17/5072 , G06F2217/70 , H03K3/0375 , H03K3/35606 , H03K3/35625
摘要： This disclosure relates generally to sequential state elements (SSEs). More specifically, embodiments of flip-flops are disclosed, along with computerized methods and systems of designing the same. In one embodiment, the flip-flop includes a substrate and subcircuits that are formed on the substrate. The subcircuits provide subfunctions, wherein each of the subcircuits provides at least one of the subfunctions. More specifically, the subfunctions are provided in a sequential logical order by the subcircuits so that the flip-flop provides a flip-flop function. However, the subcircuits are interleaved out of the sequential logical order with respect to a corresponding subfunction provided by each of the subcircuits along a vector defined by the substrate. In this manner, interleaving the subcircuits along the vector of the substrate can provide separation between charge collection nodes without requiring increases in size. Thus, the flip-flop can be more compact and less expensive to manufacture.
摘要翻译：本公开一般涉及顺序状态元素（SSEs）。更具体地，公开了触发器的实施例，以及计算机化的方法和设计它们的系统。在一个实施例中，触发器包括形成在衬底上的衬底和子电路。子电路提供子功能，其中每个子电路提供至少一个子功能。更具体地，通过子电路以顺序逻辑顺序提供子功能，使得触发器提供触发器功能。然而，子电路相对于由基板限定的矢量由每个子电路提供的相应的子功能从顺序逻辑顺序交错。以这种方式，沿着衬底的矢量交叉子电路可以提供电荷收集节点之间的间隔，而不需要增加尺寸。因此，触发器可以更紧凑并且制造成本更低。

5. 发明授权

US08420846B2 Process for producing (S)-3-[(1-dimethylamino)ethyl] phenyl-N-ethyl-N-methyl-carbamate via novel intermediates 有权
标题翻译：通过新型中间体制备（S）-3 - [（1-二甲基氨基）乙基]苯基-N-乙基-N-甲基 - 氨基甲酸酯的方法
公开(公告)号：US08420846B2
公开(公告)日：2013-04-16
申请号：US13060666
申请日：2009-08-25
申请人： Shailendra Kumar Dubey , Vikas Bansal , Kamaljeet Pannu , Sushil Kumar Dubey
发明人： Shailendra Kumar Dubey , Vikas Bansal , Kamaljeet Pannu , Sushil Kumar Dubey
IPC分类号： C07C303/28 , C07C309/73 , C07C271/42 , C07C269/00
CPC分类号： C07C309/73 , C07B2200/07 , C07C213/00 , C07C269/00 , C07C215/50 , C07C271/44
摘要： Disclosed herein are novel intermediates and process for large scale production of (S)-3-[(1-dimethylamino)ethyl]phenyl-N-ethyl-N-methyl-carbamate (rivastigmine) or its pharmaceutically acceptable salts employing the novel intermediates. Further provided are methods for producing the novel intermediates thereof.
摘要翻译：本文公开了新型中间体和用于大规模生产（S）-3 - [（1-二甲基氨基）乙基]苯基-N-乙基-N-甲基 - 氨基甲酸酯（利伐斯的明）或其药学上可接受的盐的新型中间体的方法。还提供了制备其新型中间体的方法。

6. 发明申请

US20120045592A1 Process to Deposit Diamond Like Carbon as Surface of a Shaped Object 有权
标题翻译：沉积类似碳的钻石作为形状物体表面的过程
公开(公告)号：US20120045592A1
公开(公告)日：2012-02-23
申请号：US13201210
申请日：2010-01-27
申请人： Sushil Kumar , Prakash Narain Dixit , Chandra Mohan Singh Rauthan
发明人： Sushil Kumar , Prakash Narain Dixit , Chandra Mohan Singh Rauthan
IPC分类号： C23C16/27 , C23C16/509
CPC分类号： C23C16/26 , B65D23/02 , C23C16/0272 , C23C16/045 , C23C16/45578 , C23C16/509 , H01J37/32091
摘要： A plasma based deposition process to deposit thin film on the inner surfaces of the shaped objects such as plastic or metallic object like bottles, hollow tubes etc. at room temperature has been developed. In present invention uniform hydrogenated amorphous carbon (also called Diamond-Like Carbon, DLC) films on inner surfaces of plastic bottles is successfully deposited. Applications of such product include entire food and drug industries. There is a huge demand of polyethylene terephthalate (PET) or polyethylene naphthalate (PEN)) bottles, meant for the storage of potable water, carbonated soft drinks, wines, medicines etc. However, the higher cost prohibits their wide, spread use. The cheaper alternative is to use plastic bottles inside coated with chemically inert material such as Diamond-Like Carbon (DLC) will be commercially viable. Inventor process can be scaled up for mass production. This process can also be used for coating on inner surface of metallic cane or tube with a carbide forming interlayer (like hydrogenated amorphous silicon) to get the DLC films with better adhesion to inner surface of metals.
摘要翻译：已经开发了在室温下在诸如塑料或金属物体（如瓶子，中空管等）的成形物体的内表面上沉积薄膜的等离子体沉积工艺。在本发明中，成功地沉积了塑料瓶内表面上均匀的氢化无定形碳（也称为金刚石碳，DLC）膜。这些产品的应用包括整个食品和药品行业。聚对苯二甲酸乙二醇酯（PET）或聚萘二甲酸乙二醇酯（PEN））瓶子的需求很大，用于储存饮用水，碳酸软饮料，葡萄酒，药品等。但是，更高的成本禁止其广泛使用。更便宜的替代方法是使用塑料瓶内涂覆有化学惰性材料，如金刚石碳（DLC），这在商业上是可行的。发明人流程可以扩大批量生产。该方法也可用于在金属手杖或管的内表面上涂覆碳化物形成中间层（如氢化非晶硅），以使DLC膜具有更好的金属内表面附着力。

7. 发明申请

US20110211476A1 METHOD FOR UPLINK SPECTRUM MONITORING FOR SPARSE OVERLAY TDMA SYSTEMS 有权
标题翻译：用于稀疏叠加TDMA系统的上行链路光谱监测方法
公开(公告)号：US20110211476A1
公开(公告)日：2011-09-01
申请号：US13084300
申请日：2011-04-11
申请人： Mathilde Benveniste , Sushil Kumar Prabhu
发明人： Mathilde Benveniste , Sushil Kumar Prabhu
IPC分类号： H04J3/14
CPC分类号： H04W16/14 , H04W24/00
摘要： Spectrum monitoring measurements are made by microcell base stations in a layered cellular network, while not serving calls or engaged in processing calls. The microcell base station transmits a first control message from to a microcell mobile station, to increase the duration for the mobile station to reside in the camping state on a control channel of the microcell base station. The microcell base station transmits a second control message from the microcell base station to the microcell mobile station, to increase the duration for the mobile station to reside in a call origination state while attempting to access a control channel of the microcell base station. Then, to perform the spectrum monitoring measurement, the base station's transmitter is turned off, the receiver is retuned to the frequency to be monitored, a signal strength measurement taken on that frequency, the receiver is retuned back to its assigned frequency, and the transmitter is turned back on, all in a short time interval. Because the measurement time is so short, it is possible to take spectrum-monitoring measurements without causing inactive mobiles registered on the measuring base station to reselect control channel. Mobiles initiating a call during a spectrum monitoring measurement by its base station are also delayed in their control channel reselection.
摘要翻译：频谱监视测量由分层蜂窝网络中的微蜂窝基站进行，而不提供呼叫或从事处理呼叫。微小区基站向微小区移动台发送第一控制消息，以在微小区基站的控制信道上增加移动站驻留在驻留状态的持续时间。微小区基站从微小区基站向微小区移动台发送第二控制消息，以增加移动台驻留在呼叫发起状态的持续时间，同时尝试接入微小区基站的控制信道。然后，为了执行频谱监测测量，基站的发射机被关闭，接收机被重新调谐到待监视的频率，在该频率上进行的信号强度测量，接收机被重新调回其分配的频率，并且发射机被重新打开，全部在短时间内。由于测量时间如此之短，可以进行频谱监测测量，而不会导致测量基站上登记的无效移动台重新选择控制信道。在其基站进行频谱监测测量期间发起呼叫的移动台在其控制信道重选中也被延迟。

8. 发明申请

US20110184167A1 PROCESS FOR THE PREPARATION OF TEMSIROLIMUS AND ITS INTERMEDIATES 失效
标题翻译：制备纤维素及其中间体的方法
公开(公告)号：US20110184167A1
公开(公告)日：2011-07-28
申请号：US13016235
申请日：2011-01-28
申请人： Nitin Gupta , Vishal Handa , Abir Kumar Pal , Hemant Kumar Singh , Saswata Lahiri , Sushil Kumar Dubey
发明人： Nitin Gupta , Vishal Handa , Abir Kumar Pal , Hemant Kumar Singh , Saswata Lahiri , Sushil Kumar Dubey
IPC分类号： C07D498/12 , C07D407/12
CPC分类号： C07D498/18 , C07D319/06
摘要： Novel intermediates, process for their preparation and their use in the preparation of therapeutically effective antineoplastic agents, in particular Temsirolimus of formula (I).
摘要翻译：新型中间体，其制备方法及其在制备治疗有效的抗肿瘤药物中的用途，特别是式（I）的替西罗莫司。

9. 发明授权

US07984031B2 Query builder for testing query languages 有权
标题翻译：用于测试查询语言的查询构建器
公开(公告)号：US07984031B2
公开(公告)日：2011-07-19
申请号：US12184627
申请日：2008-08-01
申请人： Sushil Kumar Chordia , Edward John Triou, Jr.
发明人： Sushil Kumar Chordia , Edward John Triou, Jr.
IPC分类号： G06F17/30
CPC分类号： G06F17/30392
摘要： Query testing is enabled across one or more query languages utilizing an abstract representation of a query. From this abstract representation, queries associated with one or more specific query languages are generated. Further, a verification scheme can be implemented for a specific store and/or query language to facilitate generation of an expected result for comparison with an actual result of test query evaluation. Further yet, data driving and/or modeling can be leveraged to further aid query testing.
摘要翻译：利用查询的抽象表示，使用一个或多个查询语言启用查询测试。从该抽象表示中，生成与一个或多个特定查询语言相关联的查询。此外，可以针对特定的存储和/或查询语言实现验证方案，以便于产生预期结果以与测试查询评估的实际结果进行比较。此外，可以利用数据驱动和/或建模来进一步帮助查询测试。

10. 发明申请

US20110065726A1 Organic Compounds 有权
标题翻译：有机化合物
公开(公告)号：US20110065726A1
公开(公告)日：2011-03-17
申请号：US12376057
申请日：2007-07-31
申请人： Zhuoliang CHEN , Sushil Kumar Sharma , Christopher Straub , Mark G. Charest , Feng He , Run-Ming David Wang , Leigh Zawel , Christine Hiu-Tung Chen , Miao Dai , Huangshu Lei , Ly Pham , Fan Yang
发明人： Zhuoliang CHEN , Sushil Kumar Sharma , Christopher Straub , Mark G. Charest , Feng He , Run-Ming David Wang , Leigh Zawel , Christine Hiu-Tung Chen , Miao Dai , Huangshu Lei , Ly Pham , Fan Yang
IPC分类号： C07D401/12 , A61P35/04 , A61K31/44 , A61K31/4439 , A61K31/427 , A61K31/422 , A61K31/506 , C07D413/12 , C07D417/12
CPC分类号： C07D417/04 , A61K31/427 , A61K45/06 , C07K5/06191
摘要： The present invention is directed to a compound of the formula: or pharmaceutically acceptable salts thereof and use of such compounds for treating proliferative diseases such as cancer, in mammals.
摘要翻译：本发明涉及下式的化合物或其药学上可接受的盐，以及在哺乳动物中用于治疗增殖性疾病例如癌症的用途。

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