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1. 发明授权

US5686484A Milbemycin derivatives, their preparation and their use 失效
标题翻译：米尔霉素衍生物，其制备及其用途
公开(公告)号：US5686484A
公开(公告)日：1997-11-11
申请号：US396662
申请日：1995-03-01
申请人： Yasuhiro Morisawa , Akio Saito , Satoru Naito , Toshimitsu Toyama , Susumu Kaneko , Louis-Pierre Molleyres , Jean-Claude Gehret
发明人： Yasuhiro Morisawa , Akio Saito , Satoru Naito , Toshimitsu Toyama , Susumu Kaneko , Louis-Pierre Molleyres , Jean-Claude Gehret
IPC分类号： A01N43/90 , C07D493/22 , C07H19/01 , A61K31/335 , C07D315/00
CPC分类号： C07D493/22 , A01N43/90 , C07H19/01
摘要： Compounds of formula (I): ##STR1## and of formula (I).sub.w : ##STR2## in which: A represents group having one of the following formulae: ##STR3## wherein R.sup.2, R.sup.3 and R.sup.4 are independently selected from the group consisting of hydrogen atoms, halogen atoms, alkyl groups having from 1 to 4 carbon atoms, and alkoxy groups having from 1 to 4 carbon atoms; R.sup.1, R.sub.w.sup.1 and R.sub.w.sup.2 are, for example, hydrogen, halogen, cyano, nitro, optically substituted alkyl, alkoxy or alkoxyalkoxy; X or X.sub.w is hydroxy, alkanoyloxy, substituted alkanoyloxy or hydroxyimino; R.sup.3.sub.w and R.sup.4.sub.w are each hydrogen, alkyl or alkoxy; R.sup.5 and R.sup.5.sub.w are methyl, ethyl, isopropyl or sec-butyl; and salts thereof have valuable anthelmintic, acaricidal and insecticidal activities.
摘要翻译：式（I）化合物：其中：A表示具有下式之一的基团：CHR 2 CHR 3 CHR 4 CR 2 CR 3 CHR 4或（I）其中R 2，R 3和R 4独立地选自氢原子，卤素原子，具有1至4个碳原子的烷基和具有1至4个碳原子的烷氧基; R1，Rw1和Rw2是例如氢，卤素，氰基，硝基，光学取代的烷基，烷氧基或烷氧基烷氧基; X或Xw是羟基，烷酰氧基，取代的烷酰氧基或羟基亚氨基; R3w和R4w各自为氢，烷基或烷氧基; R5和R5w是甲基，乙基，异丙基或仲丁基; 其盐具有宝贵的驱虫，杀螨和杀虫活性。

2. 发明授权

US5177110A Injectable parasiticidal composition 失效
标题翻译：注射杀虫剂组合物
公开(公告)号：US5177110A
公开(公告)日：1993-01-05
申请号：US689399
申请日：1991-04-22
申请人： Walter Oechslein , Jean-Claude Gehret , Ernst Hess , Sabine Rossow
发明人： Walter Oechslein , Jean-Claude Gehret , Ernst Hess , Sabine Rossow
IPC分类号： A61K9/00 , A61K31/17 , A61K31/335 , A61K31/44 , A61K31/445 , A61K31/495 , A61K31/50 , A61K31/505 , A61K31/55 , A61K47/00 , A61K47/22
CPC分类号： A61K9/0014 , A61K31/17 , A61K31/335 , A61K31/44 , A61K31/445 , A61K31/495 , A61K31/50 , A61K31/505 , A61K31/55 , A61K47/22
摘要： Parenterally injectable compositions for controlling parasites, which compositions contain from 0.1 to 10% of a benzoylurea as active ingredient, from 0.1 to 60% of a 1-substituted azacycloalkan-2-one, from 2 to 90% of a physiologically tolerable surfactant or mixture of surfactants and, if appropriate, as stabilizing component, from 0.05 to 15% of an acid or a buffer mixture and add 100% of a physiologically tolerable hydrophilic solvent or mixture of solvents or a mixture of physiologically tolerable hydrophilic and lipophilic solvents.
摘要翻译：用于控制寄生虫的肠胃外可注射组合物，该组合物含有0.1至10％的作为活性成分的苯甲酰脲，0.1至60％的1-取代的氮杂环烷-2-酮，2-90％的生理上可耐受的表面活性剂或混合物的表面活性剂，如果合适的话，作为稳定组分，0.05至15％的酸或缓冲混合物，并加入100％生理上可耐受的亲水溶剂或溶剂混合物或生理上可耐受的亲水和亲脂性溶剂的混合物。

3. 发明授权

US5132314A Anthelmintics 失效
标题翻译： ANTHELMINTICS
公开(公告)号：US5132314A
公开(公告)日：1992-07-21
申请号：US783433
申请日：1991-10-25
申请人： Peter Maienfisch , Christof Hildenbrand , Jean-Claude Gehret
发明人： Peter Maienfisch , Christof Hildenbrand , Jean-Claude Gehret
IPC分类号： A23K1/16 , A61K31/44 , A61K31/4402 , A61K31/4418 , A61K31/505 , A61P33/00 , C07D213/64 , C07D213/643 , C07D213/70 , C07D213/84 , C07D213/85 , C07D239/34 , C07D239/38 , C07D239/56
CPC分类号： C07D213/643 , C07D213/85 , C07D239/34 , C07D239/38
摘要： Anthelmintically active compounds of formula I are described ##STR1## in which R.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, C.sub.1 -C.sub.2 thioalkyl, C.sub.1 -C.sub.2 haloalkyl, nitro, C.sub.1 -C.sub.2 alkoxy, or the group SO.sub.n R in which R is C.sub.1 -C.sub.2 alkyl or phenyl and n is 0, 1 or 2;R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 haloalkoxy or C.sub.1 -C.sub.2 alkoxy;R.sub.3 is hydrogen or C.sub.1 -C.sub.2 alkyl;R.sub.4 is hydrogen or C.sub.1 -C.sub.2 alkyl;R.sub.5 is hydrogen, halogen or C.sub.1 -C.sub.5 alkyl;R.sub.6 is hydrogen, halogen or C.sub.1 -C.sub.5 alkyl;R.sub.7 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, nitro, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 haloalkoxy or C.sub.1 -C.sub.2 alkoxy;R.sub.8 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 haloalkoxy or C.sub.1 -C.sub.2 alkoxy;R.sub.9 is hydrogen, halogen, C.sub.1 -C.sub.2 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 haloalkoxy or C.sub.1 -C.sub.2 alkoxy;R.sub.10 is hydrogen, halogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 alkylthio, C.sub.3 -C.sub.6 cycloalkyl or cyano;R.sub.11 is hydrogen,halogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.2 alkylthio or C.sub.3 -C.sub.6 cycloalkyl;R.sub.12 is hydrogen or halogen; andY is .dbd.CH-- or .dbd.N--; including the physiologically tolerable acid addition salts thereof, and also the preparation and use thereof and novel intermediates.

4. 发明授权

US4954484A Parasiticides and insecticides 失效
标题翻译：杀虫剂和杀虫剂
公开(公告)号：US4954484A
公开(公告)日：1990-09-04
申请号：US172616
申请日：1988-03-24
申请人： Jean-Claude Gehret
发明人： Jean-Claude Gehret
IPC分类号： C07D493/22 , A01N43/90 , A61K31/365 , A61P33/00 , C07H19/01
CPC分类号： C07H19/01 , A01N43/90 , Y02P20/55
摘要： Novel compounds of formula ##STR1## in which A is a ##STR2## group wherein R.sub.1 is hydrogen or an OH-protecting group, and R.sub.11 is hydrogen, an OH-protecting group, or an alkyl, cycloalkyl or acyl group,R.sub.2 is methyl, ethyl, isopropyl, sec.-butyl or a --C(CH.sub.3).dbd.CH--E group wherein E is methyl, ethyl or isopropyl,R.sub.3 and R.sub.4 together represent a bond between the two carbon atoms to which they are bonded, or together represent a --C(X')(Z')-- group wherein X' and Z' each represents, independently of the other, hydrogen or halogen, andX and Z each represents, independently of the other, hydrogen or halogen,the preparation of the novel compounds and the use thereof for controlling parasites of productive livestock and for controlling harmful insects.
摘要翻译：式（Ⅰ）的新颖化合物，其中A是一个基团，其中R1是氢或OH-保护基，R11是氢，OH-保护基或烷基，环烷基或酰基， R2是甲基，乙基，异丙基，仲丁基或-C（CH 3）= CH-E基团，其中E是甲基，乙基或异丙基，R 3和R 4一起代表它们所键合的两个碳原子之间的键或者一起表示-C（X'）（Z'） - 基团，其中X'和Z'各自独立地表示氢或卤素，X和Z各自独立地表示氢或卤素，新化合物的制备及其用于控制生产性家畜寄生虫和控制有害昆虫的用途。

5. 发明授权

US4857509A 13.beta.-alkylmilbemycin derivatives for controlling parasites of animals and plants 失效
标题翻译： 13个β-烷基米比霉素衍生物，用于控制动物和植物的寄生虫
公开(公告)号：US4857509A
公开(公告)日：1989-08-15
申请号：US820490
申请日：1986-01-17
申请人： Bruno Frei , Anthony C. O'Sullivan , Jean-Claude Gehret
发明人： Bruno Frei , Anthony C. O'Sullivan , Jean-Claude Gehret
IPC分类号： A01N43/90 , A01N55/00 , A61K31/35 , A61K31/365 , A61K31/695 , A61K31/70 , A61K31/7042 , A61K31/7048 , A61P33/00 , A61P33/10 , C07D493/22 , C07F7/18 , C07H17/08 , C07H19/01
CPC分类号： C07H19/01 , A01N43/90 , A01N55/00
摘要： The invention relates to parasiticidally and insecticidally highly active compounds of formula I ##STR1## wherein R is C.sub.1 -C.sub.10 alkyl;R.sub.1 is hydrogen, a silyl group or a sugar residue; andR.sub.2 is methyl, ethyl, isopropyl or sec-butyl, and to the preparation thereof starting from suitably substituted 15-ester or 13.beta.-ester milbemycins.
摘要翻译：本发明涉及杀虫活性和杀虫活性高的式I化合物（Ⅰ），其中R是C1-C10烷基; R1是氢，甲硅烷基或糖残基; 并且R 2是甲基，乙基，异丙基或仲丁基，并且从适当取代的15-酯或13β-甲酯米尔倍霉素开始制备。

6. 发明授权

US4855317A Insecticides and parasiticides 失效
标题翻译：杀虫剂和杀寄生虫剂
公开(公告)号：US4855317A
公开(公告)日：1989-08-08
申请号：US160237
申请日：1988-02-25
申请人： Jean-Claude Gehret
发明人： Jean-Claude Gehret
IPC分类号： C07D493/22 , A01N43/90 , A61K31/365 , A61P33/00 , C07H19/01
CPC分类号： C07H19/01 , A01N43/90 , Y02P20/55
摘要： The present invention relates to novel C(29)-oximinomilbemycin derivatives of formula I, to their preparation and to the use thereof for controlling pests. The invention further relates to pesticidal compositions which contain at least one of these compounds as active ingredient.The novel compounds have the general formula I ##STR1## wherein X is a group selected from --CH(OR.sub.1)--, --C(O)-- or --C(.dbd.N--OR)--,R.sub.1 is hydrogen or a OH protective group,R is hydrogen, a OH protective group, an alkyl, cycloalkyl or acyl group,R.sub.2 is methyl, ethyl, isopropyl, sec-butyl or the ##STR2## wherein A is methyl, ethyl or isopropyl; and R.sub.3 is hydrogen, C.sub.1 -C.sub.6 alkyl, C.sub.2 -C.sub.6 alkenyl, a radial selected from the group consisting of phenyl and benzyl which is unsubstituted or substituted by one or more members selected from the group consisting of halogen, C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 alkylthio, C.sub.1 -C.sub.3 haloalkyl, nitro or cyano, or is the group U ##STR3## wherein n is 0, 1, 2, 3, 4 or 5, E is oxygen or --CH(R.sub.d)-- and R.sub.z is hydrogen, R.sub.a is hydrogen, halogen, C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkoxy or 2-tetrahydropyranyl, and R.sub.b, R.sub.c and R.sub.d are each independently hydrogen, halogen, C.sub.1 -C.sub.3 alkyl or C.sub.1 -C.sub.3 alkoxy, which group U may also be in unsaturated form.
摘要翻译：本发明涉及式I的新型C（29） - 阿立米尔霉素衍生物及其制备及其用于防治害虫的用途。本发明还涉及含有这些化合物中的至少一种作为活性成分的杀虫组合物。新化合物具有通式I（I）其中X是选自-CH（OR 1） - ， - C（O） - 或-C（= N-OR） - ，R 1是氢或 OH保护基，R为氢，OH保护基，烷基，环烷基或酰基，R2为甲基，乙基，异丙基，仲丁基或其中A为甲基，乙基或异丙基; 并且R 3是氢，C 1 -C 6烷基，C 2 -C 6烯基，选自苯基和苄基的放射线，其是未取代的或被一个或多个选自卤素，C 1 -C 3烷基，C 1 -C 3烷氧基， C 1 -C 3烷硫基，C 1 -C 3卤代烷基，硝基或氰基，或其中n为0,1,2,3,4或5的基团，其中E为氧或-CH（R d） - ，R z 是氢，R a是氢，卤素，C 1 -C 3烷基，C 1 -C 3烷氧基或2-四氢吡喃基，R b，R c和R d各自独立地是氢，卤素，C 1 -C 3烷基或C 1 -C 3烷氧基，U基也可以是不饱和的形成。

7. 发明授权

US4567190A Pesticidal phenylhydrazonopyrrolidines 失效
标题翻译：杀虫剂苯肼基吡咯烷
公开(公告)号：US4567190A
公开(公告)日：1986-01-28
申请号：US622826
申请日：1984-06-21
申请人： Jean-Claude Gehret , Walter Traber
发明人： Jean-Claude Gehret , Walter Traber
IPC分类号： A01N43/40 , A01N43/78 , A01N57/32 , C07D401/12 , C07D417/12 , C07F9/572 , A61K31/44
CPC分类号： C07D401/12 , A01N43/40 , A01N43/78 , A01N57/32 , C07D417/12 , C07F9/5721
摘要： Substituted phenylhydrazonopyrrolidine derivatives of the formula ##STR1## wherein R is halogen or C.sub.1 -C.sub.4 -alkyl,n is zero, 1 or 2, andR* is the group --CH.dbd.N--R.sub.1 or ##STR2## in which R.sub.1 is a pyridine group which is bound by way of a carbon atom, and which is unsubstituted or substituted by a methyl group, or is a 2-thiazolyl group, andR.sub.2 is methyl or ethyl,R.sub.3 is C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.2 -alkoxy or C.sub.1 -C.sub.4 -alkylthio, andX is oxygen or sulfur,have valuable properties for controlling pests, such as phytoparasitic and zooparasitic insects and acarids, including in particular ectoparasites.
摘要翻译：取代的苯并腙基吡咯烷衍生物，其中R是卤素或C 1 -C 4 - 烷基，n是0,1或2，R *是基团-CH = N-R 1或者其中R 1是吡啶通过碳原子结合的基团，其未被取代或被甲基取代，或是2-噻唑基，R2是甲基或乙基，R3是C1-C4-烷基，C1-C2-烷氧基或C 1 -C 4 - 烷硫基，且X为氧或硫，具有用于防治害虫的有价值的性质，例如植物寄生虫和动物寄生昆虫和螨，包括特别是外寄生虫。

8. 发明授权

US4455438A Cyclobutanone oximes 失效
标题翻译：环丁酮肟
公开(公告)号：US4455438A
公开(公告)日：1984-06-19
申请号：US376988
申请日：1982-05-10
申请人： Laurenz Gsell , Jean-Claude Gehret
发明人： Laurenz Gsell , Jean-Claude Gehret
IPC分类号： A01N47/24 , C07C131/00
CPC分类号： A01N47/24
摘要： Cyclobutanone oxime carbamates of the formula ##STR1## wherein n is 1 to 5 and X.sub.1 is hydrogen, halogen, C.sub.1 -C.sub.4 alkoxy or C.sub.1 -C.sub.4 alkylthio. A process for obtaining the compounds of the formula I and their use in pest control as well as the cyclobutanone oximes used as intermediates are described.
摘要翻译：式（I）的环丁酮肟氨基甲酸酯，其中n为1至5，X 1为氢，卤素，C 1 -C 4烷氧基或C 1 -C 4烷硫基。描述了获得式I化合物及其在病虫害防治中的用途以及用作中间体的环丁酮肟的方法。

9. 发明授权

US4946854A 3-aminobenzoylphenylureas useful for controlling parasites and insects that attack domestic animals and livestock 失效
标题翻译： 3-氨基苯甲酰苯胺可用于控制攻击家畜和牲畜的寄生虫和昆虫
公开(公告)号：US4946854A
公开(公告)日：1990-08-07
申请号：US280061
申请日：1988-12-05
申请人： Peter Maienfisch , Jean-Claude Gehret , Bruno Frei
发明人： Peter Maienfisch , Jean-Claude Gehret , Bruno Frei
IPC分类号： C07D213/64 , A01N47/34 , C07C67/00 , C07C233/58 , C07C233/65 , C07C241/00 , C07C265/16 , C07D213/643 , C07D213/70 , C07D213/74
CPC分类号： C07D213/643 , C07C233/58 , C07C265/16 , C07D213/70 , C07D213/74
摘要： Novel compounds of formula I ##STR1## wherein each of R.sup.1, R.sup.2, R.sup.3, R.sup.7, R.sup.8 and R.sup.9, independently of the others, is H or halogen,R.sup.4 is H, R.sup.10 CO-- or R.sup.11 NHCO-- wherein R.sup.10 is a C.sub.1 -C.sub.4 alkyl group which is unsubstituted or substituted by one to three identical or different substituents selected from the group consisting of halogen, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 - acyloxy and --COOG, wherein G is H, an alkali metal cation or an alkaline earth metal cation, and R.sup.11 is an unsubstituted or halo-substituted C.sub.1 -C.sub.4 alkyl or phenyl group,each of R.sup.5 and R.sup.6, independently of the other, is H, halogen, alkyl or haloalkyl andX is O, S(O)n or NH wherein n is 0, 1 or 2, the preparation of the novel compounds and their use against parasites in and on productive livestock and against insect pests, and novel starting materials and their preparation.
摘要翻译：式I的新型化合物其中R 1，R 2，R 3，R 7，R 8和R 9各自独立地为H或卤素，R 4为H，R 10 CO-或R 11 NHCO-，其中R 10为C 1 -C 1-4烷基，其被未取代或被一至三个相同或不同的选自卤素，C 1 -C 4烷氧基，C 1 -C 4 - 酰氧基和-COOG的取代基取代，其中G为H，碱金属阳离子或碱土金属金属阳离子，R11为未取代或卤素取代的C1-C4烷基或苯基，R5和R6各自独立地为H，卤素，烷基或卤代烷基，X为O，S（O）n或NH 其中n为0,1或2，新化合物的制备及其在生产性家畜和害虫中的寄生虫的用途，以及新的起始原料及其制备方法。

10. 发明授权

US4559357A Insecticidal and acaricidal phenylhydrazono- and phenylhydrazino-pyrrolidines 失效
标题翻译：杀虫和杀螨苯肼和苯肼基吡咯烷
公开(公告)号：US4559357A
公开(公告)日：1985-12-17
申请号：US501456
申请日：1983-06-06
申请人： Jean-Claude Gehret , Walter Traber
发明人： Jean-Claude Gehret , Walter Traber
IPC分类号： A01N43/36 , A01N47/36 , A01N47/38 , C07D207/22 , C07D207/14
CPC分类号： C07D207/22 , A01N43/36 , A01N47/36 , A01N47/38
摘要： Compounds of the formula ##STR1## and of the isomeric formulae ##STR2## wherein R is alkyl or halogen, R.sub.1 is hydrogen, optionally substituted alkyl or optionally substituted alkenyl, R.sub.2 is hydrogen or methyl, R.sub.3 is hydrogen, alkyl or alkenyl, and X is oxygen or sulfur, including their acid salts, are insecticidally and acaricidally active.
摘要翻译：其中R是烷基或卤素，R 1是氢，任选取代的烷基或任选被取代的链烯基，R 2是（Ⅰa）化合物及其异构体式氢或甲基，R3是氢，烷基或烯基，X是氧或硫，包括它们的酸盐，具有杀虫和杀螨活性。

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