专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 发明授权

US3846409A 10,11-METHANO 5H-DIBENZ {8 b,f{9 {0 AZEPINES 5-PHENACYL DERIVATIVES 失效
标题翻译： 10,11-甲基-5H-二苯并[b，f {9 {0，AZEPINES 5-PHENACYL DERIVATIVES
公开(公告)号：US3846409A
公开(公告)日：1974-11-05
申请号：US20574171
申请日：1971-12-07
申请人： SYNTEX INC
发明人： MARX M
IPC分类号： C07C49/80 , C07D41/08
CPC分类号： C07C49/80
摘要： Phenacyl, and ring substituted phenacyl, derivatives of 10,11dihydro-10,11-methano (and 10a-halo substituted-10,11-methano)-5( gamma -alkyl-aminopropyl)-5H-dibenz(b,f)azepine, at the N-amino side chain, and methods of preparing these compounds. The compounds are broadly prepared by treating the corresponding parent compound with omega -bromoacetophenone, or the desired ring substituted omega -bromoacetophenone. The compounds have utility for palliating conditions of mental depression, occurring in mammals related to the central nervous system.
摘要翻译：苯甲酰基和环取代的苯甲酰甲基，10,11-二氢-10,11-亚甲基（和10a-卤素取代-10,11-亚甲基）-5-（γ-烷基 - 氨基丙基）-5H-二苯并[b， f]吖庚因，N-氨基侧链和制备这些化合物的方法。通过用ω-溴苯乙酮或所需的环取代的ω-溴苯乙酮处理相应的母体化合物来广泛制备这些化合物。这些化合物可用于缓解与中枢神经系统相关的哺乳动物发生的精神抑郁症状况。

2. 发明授权

US3833559A Dibenzocycloheptenyl lactamimides 失效
标题翻译：二苯甲酰胆碱酯酶
公开(公告)号：US3833559A
公开(公告)日：1974-09-03
申请号：US32128873
申请日：1973-01-05
申请人： RICHARDSON MERRELL INC
发明人： GRISAR M , MAC KENZIE R
IPC分类号： C07D223/12 , A61K31/395 , A61K31/445 , A61K31/55 , A61P7/02 , A61P7/10 , A61P29/00 , C07D207/22 , C07D211/72 , C07D225/02 , C07D227/10 , C07D27/04 , C07D29/28 , C07D41/08
CPC分类号： C07D227/10 , Y10S514/822 , Y10S514/869
摘要： NOVEL DIBENZOCYCLOHEPTENYL LACTAMIMIDES OF THE FOLLOWING FORMULA AND PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS THEREOF ARE USEFUL AS DIURETIC AGENTS, ANTIINFLAMMATORY AGENTS, AND AS ANTICOAGULANTS.

5-(-N=C
TENE

IN THE ABOVE FORMULA N REPRESENTS AN INTEGER OF FROM 3 TO 11.

3. 发明授权

US3792042A Dihydrodibenzo(b,f)azepine derivatives 失效
标题翻译：二氢苯并（B，F）亚胺衍生物
公开(公告)号：US3792042A
公开(公告)日：1974-02-12
申请号：US3792042D
申请日：1970-06-22
申请人： RHONE POULENC SA
发明人： FOUCHE J , LEGER A
IPC分类号： A01N43/46 , A01N47/18 , C07D223/22 , C07D41/08
CPC分类号： C07D223/22 , A01N47/18
摘要： NEW 10,11-DIHYDRODIBENZO (B,F)AZEPINES OF THE FORMULA:

5-R,10-(R1-OOC-NH-)-10,11-DIHYDRO-5H-DIBENZ(B,F)AZEPINE

WHEREIN R REPRESENTS HYDROGEN OR ALKYL OF 1 THROUGH 5 CARBON ATOMS, AND R1 REPRESENTS ALKYL OF 1 THROUGH 7 CARBON ATOMS, ARE USEFUL FUNGICIDES.

4. 发明授权

US3766170A 3-benzazepines and salts thereof 失效
标题翻译： 3-BENZAZEPINES和SALTS OF
公开(公告)号：US3766170A
公开(公告)日：1973-10-16
申请号：US3766170D
申请日：1971-03-25
申请人： BOEHRINGER SOHN INGELHEIM
发明人： MENTRUP A , SCHROMM K , RENTH E , REICHL R
IPC分类号： C07D223/16 , C07D41/08
CPC分类号： C07D223/16 , Y10S514/91
摘要： COMPOUNDS OF THE FORMULA

7-(R1-CO-),R2,R3-2,3,4,5-TETRAHYDRO-1H-3-BENZAZEPINE

WHEREIN R1 IS ALKYL OF 1 TO 6 CARBON ATOMS OR TRIFLUOROMETHYL, AND R2 AND R3, WHICH MAY BE IDENTICAL TO OR DIFFERENT FROM EACH OTHER, ARE EACH HYDROGEN OR METHYL, AND NON-TOXIC, PHARMACOLOGICALLY ACCEPTABLE ACID ADDITION SALTS THEREOF; THE COMPOUNDS AS WELL AS THEIR SALTS ARE USEFUL AS APPETITE-CURBERS.

5. 发明授权

US3652588A 6-alkyl-1 2 3 4 5 6-hexahydroazepino(4 5-b)indoles 失效
标题翻译： 6-ALKYL-1 2 3 4 5 6-HEXAHYDROAZEPINO（4 5-B）吲哚
公开(公告)号：US3652588A
公开(公告)日：1972-03-28
申请号：US3652588D
申请日：1969-10-23
申请人： UPJOHN CO
发明人： HESTER JACKSON B JR
IPC分类号： C07D487/04 , C07D27/54 , C07D41/08
CPC分类号： C07D487/04
摘要： A 6-ALKYL - 1,2,3,4,5,6 - HEXAHYDROAZEPINO (4,5-B) INDOLE HAVING A SEDATIVE TRANQUILIZING AND ANOREXIGENIC ACTION OF THE FORMULA:

3-R2,6-R1,R,R''-1,2,3,4,5,6,-HEXAHYDROAZEPINO(4,5-B)INDOLE

WHEREIN R AND R'' ARE SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, ALKOXY AND ALKYL CONTAINING FROM 1 TO 3 CARBON ATOMS, INCLUSIVE, AND HALOGEN; WHEREIN R1 IS ALKYL DEFINED AS ABOVE; AND WHEREIN R2 IS SELECTED FROM THE GROUP CONSISTING OF HYDROGEN, METHYL, ETHYL, PROPYL, ALKANOYL GROUPS CONTAINING 1 TO 3 CARBON ATOMS, INCLUSIVE, BENZYL AND BENXOYL, AND THE ORGANIC AND INORGANIC ACID ADDITION SALTS OF THOSE COMPOUNDS WHEREIN >N-R2 IS AN AMINO MOIETY, INCLUDING PHARMACOLOGICALLY ACCEPTABLE ACID ADDITION SALTS OF THOSE COMPOUNDS, ARE PREPARED. THE COMPOUNDS ARE USED TO TRANQUILIZE AND SEDATE MAMMALS OR SUPPRESS HUNGER IN MAMMALS.

6. 发明授权

US3652543A Process for the production of 1 2 4 5-tetrahydro-3-azepines 失效
标题翻译：生产1 2 4 5-四氢-3-氨基辛酸的方法
公开(公告)号：US3652543A
公开(公告)日：1972-03-28
申请号：US3652543D
申请日：1968-02-15
申请人： GEIGY CHEM CORP
发明人： HOEGERLE KARL
IPC分类号： C07D203/08 , C07D223/16 , C07D41/08
CPC分类号： C07D203/08 , C07D223/16
摘要： PROCESS FOR THE PRODUCTION OF 1,2,4,5-TETRAHYDRO-3-AZEPINES FROM STYRENE VIA N-AZIRIDINYL-ALKYL-BENZENES, AND HALOGENO-ALKYLAMINO-ALKYL-BENZENES, WHICH LATTER INTERMEDIATES ARE USEFUL AS HERBICIDES; FROM THE LATTER, THE CORRESPONDING 1,2,4,5-TETRAHYDRO-3-AZEPINES ARE OBTAINED IN A SIMPLE, INDUSTRIALLY APPLICABLE PROCESS AND IN VERY SATISFACTORY YIELDS. 1,2,4,5-TETRAHYDROAZEPINES ARE USEFUL AS INTERMEDIATES IN THE PRODUCTION OF ANTIHYPERTENSIVE AGENTS, HYPOGLYCEMIC AGENTS AND SOME POSSESS THEMSELVES ANOREXOGENIC PROPERTIES.

7. 发明授权

US3642775A 10-oxo-10 11-dihydro-dibenzazepine derivative 失效
标题翻译： 10-OXO-10 11-二氢 - 二苯甲酮衍生物
公开(公告)号：US3642775A
公开(公告)日：1972-02-15
申请号：US3642775D
申请日：1970-03-04
申请人： CIBA GEIGY CORP
发明人： SCHINDLER WALTER
IPC分类号： C07D223/28 , C07D41/08
CPC分类号： C07D223/28
摘要： 10 - OXO - 10,11-DIHYDRO-5H-DIBENZ(B,F)AZEPINE-5-CARBOXAMIDE HAS A DEPRESSANT EFFECT ON THE CENTRAL NERVOUS SYSTEM; THE COMPOUNDS IS THE ACTIVE INGREDIENT OF PHARMACEUTICAL COMPOSITIONS AND IS USEFUL FOR THE TREATMENT OF PYSCHOSOMATIC DISTURBANCES, OF EPILEPSY AND OF TRIGEMINAL NEURALGIA.
摘要翻译： 10-氧代-10,11-二氢-5H-二苯并[b，f]吖庚因-5-甲酰胺对中枢神经系统具有抑制作用; 该化合物是药物组合物的活性成分，可用于治疗心身障碍，癫痫和三叉神经痛。

8. 发明授权

US3637661A 10-hydroxy-10 11-dihydro-dibenzazepine derivative 失效
标题翻译： 10-羟基-10,11-二氢 - 二苯甲酮衍生物
公开(公告)号：US3637661A
公开(公告)日：1972-01-25
申请号：US3637661D
申请日：1970-03-04
申请人： CIBA GEIGY CORP
发明人： SCHINDLER WALTER
IPC分类号： C07D223/28 , C07D41/08
CPC分类号： C07D223/28
摘要： 10 - HYDROXY - 10,11 - DIHYDRO-5H - DIBENZ(B,F)AZEPINE-5-CARBOXAMIDE HAS A DEPRESSANT EFFECT ON THE CENTRAL NERVOUS SYSTEM; THE COMPOUND IS THE ACTIVE INGREDIENT OF PHARMACEUTICAL COMPOSITIONS AND IS USEFUL FOR THE TREATMENT OF PSYCHOSOMATIC DISTURBANCES, OF EPILEPSY AND OF TRIGEMINAL NEURALGIA.

9. 发明授权

US3609138A 1-aryl-3-benzazepines 失效
标题翻译： 1-ARYL-3-BENZAZEPINES
公开(公告)号：US3609138A
公开(公告)日：1971-09-28
申请号：US3609138D
申请日：1967-12-22
申请人： CIBA GEIGY CORP
发明人： MULL ROBERT PAUL , STEVENS GEORGE DE
IPC分类号： C07D223/16 , C07D41/08
CPC分类号： C07D223/16
摘要： 3-Aliphatically substituted 1-aryl-1,2-dihydro- or 1,2,4,5tetrahydro-3-benzazepines, e.g. those of the formula

D R A W I N G

10. 发明授权

US3544557A Benzhydryl ethers 失效
标题翻译： BENZHYDRYL ETHERS
公开(公告)号：US3544557A
公开(公告)日：1970-12-01
申请号：US3544557D
申请日：1967-08-04
申请人： KONINKLIJKE PHARMA FAB NV
发明人： NAUTA WIJBE T
IPC分类号： C07D295/088 , C07D41/08
CPC分类号： C07D295/088 , Y10S514/818 , Y10S514/929

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式