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1. 发明授权

US11284620B2 Picolinamide compounds with fungicidal activity 有权
公开(公告)号：US11284620B2
公开(公告)日：2022-03-29
申请号：US16722451
申请日：2019-12-20
申请人： CORTEVA AGRISCIENCE LLC
发明人： Karla Bravo-Altamirano , Yu Lu , Brian A. Loy , Zachary A. Buchan , David M. Jones , Jeremy Wilmot , Jared W. Rigoli , Kyle A. Dekorver , John F. Daeuble , Jessica Herrick , Xuelin Wang , Chenglin Yao , Kevin G. Meyer
IPC分类号： A01N47/12 , A01N43/40 , A01N43/10 , A01N37/44 , A01N25/00 , C07D313/00 , A01N43/16 , C07C229/08 , C07C229/20 , C07C229/22 , C07C235/52 , C07C271/22 , C07D213/81 , C07D311/82 , C07D333/16 , C07D405/12 , C07D409/14 , A01P3/00
摘要： This disclosure relates to picolinamides of Formula I and their use as fungicides.

2. 发明授权

US10590066B2 Biocompositions for 3D printing 有权
公开(公告)号：US10590066B2
公开(公告)日：2020-03-17
申请号：US16110639
申请日：2018-08-23
申请人： 3D-BIOMATERIALS, LLC
发明人： Sajal Das , Patrick Shipman , Scott Shuler
IPC分类号： C07C233/46 , C08L33/10 , C08L77/12 , C08L67/06 , C07C235/52 , C08F220/36 , C07C235/34 , A61L27/18 , C07C271/22 , C07C237/22 , C08F220/60 , C07C237/20 , A61K9/00 , B33Y70/00
摘要： The present disclosure is directed to resins and to polymers, copolymers, and blends formed therefrom.

3. 发明授权

US10588318B2 Picolinamide compounds with fungicidal activity 有权
公开(公告)号：US10588318B2
公开(公告)日：2020-03-17
申请号：US15953394
申请日：2018-04-13
申请人： Dow AgroSciences LLC
发明人： Karla Bravo-Altamirano , Yu Lu , Brian A. Loy , Zachary A. Buchan , David M. Jones , Jeremy Wilmot , Jared W. Rigoli , Kyle A. Dekorver , John F. Daeuble, Sr. , Jessica Herrick , Xuelin Wang , Chenglin Yao , Kevin G. Meyer
IPC分类号： A01N47/12 , A01N43/40 , A01N43/10 , A01N37/44 , A01N25/00 , C07D313/00 , A01N43/16 , C07C229/08 , C07C229/20 , C07C229/22 , C07C235/52 , C07C271/22 , C07D213/81 , C07D311/82 , C07D333/16 , C07D405/12 , C07D409/14
摘要： This disclosure relates to picolinamides of Formula I and their use as fungicides.

4. 发明申请

US20200046738A1 FATTY ACID ACETYLATED SALICYLATES AND THEIR USES 审中-公开
公开(公告)号：US20200046738A1
公开(公告)日：2020-02-13
申请号：US16353575
申请日：2019-03-14
申请人： Catabasis Pharmaceuticals, Inc.
发明人： Jill C. Milne , Michael R. Jirousek , Jean E. Bemis , Jesse J. Smith
IPC分类号： A61K31/609 , C07C69/86 , C07C69/94 , C07C233/18 , C07C233/49 , C07C237/22 , C07C271/28 , C07C275/42 , C07D295/182 , C07D295/192 , C07C233/55 , C07C235/60 , C07C235/52
摘要： The invention relates to Fatty Acid Acetylated Salicylate Derivatives; compositions comprising an effective amount of a Fatty Acid Acetylated Salicylate Derivative; and methods for treating or preventing an inflammatory disorder comprising the administration of an effective amount of a Fatty Acid Acetylated Salicylate Derivative.

5. 发明申请

US20190010129A1 Amide derivatives as lysophosphatidic acid receptor antagonists 审中-公开
公开(公告)号：US20190010129A1
公开(公告)日：2019-01-10
申请号：US15999570
申请日：2018-08-20
申请人： Takeda Pharmaceutical Company Limited
发明人： William Buffham , Hannah Canning , Richard Davenport , William Farnaby , Stephen Mack , Alka Parmar , Susanne Wright
IPC分类号： C07D239/34 , C07C255/54 , A61K31/44 , A61K31/505 , C07C235/44 , C07D213/81 , A61K31/277 , C07D213/78 , C07C235/46 , C07C235/52 , A61K31/195
摘要： The present invention provides compounds of formula (I) and pharmaceutically acceptable salts thereof, formula (I) wherein R1, X, m, R2, Y, R3, Z, n, R4, A and B are as defined in the specification, processes for their preparation, pharmaceutical compositions containing them and their use in therapy.

6. 发明申请

US20170295792A1 USE OF PICOLINAMIDE COMPOUNDS AS FUNGICIDES 审中-公开
公开(公告)号：US20170295792A1
公开(公告)日：2017-10-19
申请号：US15036316
申请日：2015-12-18
申请人： DOW AGROSCIENCES LLC
发明人： Karla BRAVO-ALTAMIRANO , Yu LU , Brian A. LOY , Zachary A. BUCHAN , David M. JONES , Jeremy WILMOT , Jared W. RIGOLI , Kyle A. DEKORVER , John F. DAEUBLE, Sr. , Jessica HERRICK , Xuelin WANG , Chenglin YAO , Kevin G. MEYER
IPC分类号： A01N47/12 , C07D405/12 , C07D333/16 , C07D311/82 , C07D213/81 , C07C271/22 , A01N37/44 , C07C229/22 , C07C229/20 , C07C229/08 , A01N43/40 , A01N43/16 , A01N43/10 , C07C235/52 , C07D409/14
CPC分类号： A01N47/12 , A01N25/00 , A01N37/44 , A01N43/10 , A01N43/16 , A01N43/40 , C07C229/08 , C07C229/20 , C07C229/22 , C07C235/52 , C07C271/22 , C07D213/81 , C07D311/82 , C07D313/00 , C07D333/16 , C07D405/12 , C07D409/14
摘要： This disclosure relates to picolinamides of Formula I and their use as fungicides.

7. 发明申请

US20050256116A1 Novel biaromatic compounds which activate PPARy type receptors and cosmetic/pharmaceutical compositions comprised thereof 失效
标题翻译：活化PPARγ型受体的新型双芳族化合物和包含它们的化妆品/药物组合物
公开(公告)号：US20050256116A1
公开(公告)日：2005-11-17
申请号：US11131302
申请日：2005-05-18
申请人： Laurence Clary , Claire Bouix-Peter , Michel Rivier , Pascal Collette , Andre Jomard
发明人： Laurence Clary , Claire Bouix-Peter , Michel Rivier , Pascal Collette , Andre Jomard
IPC分类号： A61K8/44 , A61K8/49 , A61K31/165 , A61K31/195 , A61K31/4015 , A61K31/4245 , A61K31/537 , A61Q5/00 , A61Q19/00 , A61Q19/08 , C07C229/36 , C07C233/47 , C07C233/54 , C07C233/55 , C07C233/65 , C07C233/87 , C07C235/52 , C07C235/60 , C07C235/74 , C07C235/84 , C07C237/20 , C07C237/40 , C07C243/28 , C07C271/22 , C07C275/42 , C07C323/60 , C07C335/22 , C07D207/26 , C07D207/27 , C07D207/32 , C07D207/335 , C07D211/34 , C07D211/62 , C07D213/38 , C07D213/40 , C07D263/32 , C07D271/06 , C07D271/10 , C07D295/088 , C07D295/185 , C07D295/205 , C07D307/81 , C07D333/20
CPC分类号： C07D207/27 , A61K8/44 , A61K8/49 , A61Q5/00 , A61Q19/00 , A61Q19/08 , C07C229/36 , C07C233/47 , C07C233/54 , C07C233/55 , C07C233/65 , C07C233/81 , C07C233/87 , C07C235/52 , C07C235/60 , C07C235/74 , C07C235/84 , C07C237/20 , C07C237/40 , C07C243/28 , C07C271/22 , C07C275/42 , C07C323/60 , C07C335/22 , C07C2601/02 , C07C2601/14 , C07D207/335 , C07D211/16 , C07D211/34 , C07D211/62 , C07D213/38 , C07D213/40 , C07D263/32 , C07D265/30 , C07D271/06 , C07D271/10 , C07D295/088 , C07D295/185 , C07D295/205 , C07D307/81 , C07D333/20
摘要： Novel biaromatic compounds having the structural formula (I) below: are formulated into pharmaceutical compositions suited for administration in human or veterinary medicine (in dermatology, and also in the fields of cardiovascular diseases, immune diseases and/or diseases associated with lipid metabolism), or, alternatively, into cosmetic compositions.
摘要翻译：具有下述结构式（I）的新颖的双芳族化合物被配制成适用于人或兽医药物（皮肤病学以及与心血管疾病，免疫疾病和/或脂质代谢相关的疾病领域）的药物组合物，或替代地，进入化妆品组合物。

8. 发明申请

US20050059705A1 Aryl and heteroaryl compounds, compositions, and methods of use 失效
标题翻译：芳基和杂芳基化合物，组合物和使用方法
公开(公告)号：US20050059705A1
公开(公告)日：2005-03-17
申请号：US10913168
申请日：2004-08-06
申请人： Adnan Mjalli , Robert Andrews , Xiao-Chuan Guo , Daniel Christen , Devi Gohimmukkula , Guoxiang Huang , Robert Rothlein , Sameer Tyagi , Tripura Yaramasu , Christopher Behme
发明人： Adnan Mjalli , Robert Andrews , Xiao-Chuan Guo , Daniel Christen , Devi Gohimmukkula , Guoxiang Huang , Robert Rothlein , Sameer Tyagi , Tripura Yaramasu , Christopher Behme
IPC分类号： A61P31/12 , C07C233/87 , C07C235/42 , C07C235/52 , C07C235/60 , C07C235/66 , C07C237/36 , C07C237/42 , C07C271/20 , C07C311/08 , C07C311/09 , C07C311/21 , C07C311/44 , C07C317/32 , C07C323/36 , C07D295/155 , C07D41/02 , A61K31/4439 , C07D43/02
CPC分类号： C07D295/155 , C07C233/87 , C07C235/42 , C07C235/52 , C07C235/60 , C07C235/66 , C07C237/36 , C07C237/42 , C07C271/20 , C07C311/08 , C07C311/09 , C07C311/21 , C07C311/44 , C07C317/32 , C07C323/36 , C07C2601/08
摘要： This invention provides aryl and heteroaryl compounds, methods of their preparation, pharmaceutical compositions comprising the compounds, and their use in treating human or animal disorders. The compounds of the invention may be antagonists, or partial antagonist of factor IX and/or factor XI and thus, may be useful for inhibiting the intrinsic pathway of blood coagulation. The compounds may be useful in a variety of applications including the management, treatment and/or control of diseases caused in part by the intrinsic clotting pathway.
摘要翻译：本发明提供芳基和杂芳基化合物，其制备方法，包含该化合物的药物组合物及其在治疗人或动物病症中的用途。本发明的化合物可以是拮抗剂或因子IX和/或因子XI的部分拮抗剂，因此可用于抑制凝血的内在途径。所述化合物可用于各种应用，包括部分由内在凝血途径引起的疾病的管理，治疗和/或控制。

9. 发明申请

US20050049310A1 Aryl and heteroaryl compounds, compositions and methods of use 失效
标题翻译：芳基和杂芳基化合物，组合物和使用方法
公开(公告)号：US20050049310A1
公开(公告)日：2005-03-03
申请号：US10913882
申请日：2004-08-06
申请人： Adnan Mjalli , Guoxiang Huang , Murty Arimilli , Thomas Yokum , Jeff Zhu
发明人： Adnan Mjalli , Guoxiang Huang , Murty Arimilli , Thomas Yokum , Jeff Zhu
IPC分类号： A61P31/12 , C07C233/87 , C07C235/42 , C07C235/52 , C07C235/60 , C07C235/66 , C07C237/36 , C07C237/42 , C07C271/20 , C07C311/08 , C07C311/09 , C07C311/21 , C07C311/44 , C07C317/32 , C07C323/36 , C07D295/155 , A61K31/195 , A61K31/137 , A61K31/15
CPC分类号： C07D295/155 , C07C233/87 , C07C235/42 , C07C235/52 , C07C235/60 , C07C235/66 , C07C237/36 , C07C237/42 , C07C271/20 , C07C311/08 , C07C311/09 , C07C311/21 , C07C311/44 , C07C317/32 , C07C323/36 , C07C2601/08
摘要： This invention provides aryl and heteroaryl compounds of Formula (I) as described herein, and methods of their preparation. Also provided are pharmaceutical compositions made with the compounds of Formula (I) and methods for making such compositions. The compounds of Formula (I) may activate an erythropoietin receptor and thus, may be useful to induce red blood cell production. The compounds of Formula (I) and compositions including compounds of Formula (I) may be useful in a variety of applications including the management, treatment and/or control of diseases caused at least in part by deficient (or inefficient) EPO production relative to hemoglobin level.
摘要翻译：本发明提供了本文所述的式（I）的芳基和杂芳基化合物及其制备方法。还提供了用式（I）的化合物制备的药物组合物和制备这些组合物的方法。式（I）的化合物可以激活促红细胞生成素受体，因此可用于诱导红细胞生成。式（I）化合物和包含式（I）化合物的组合物可用于各种应用，包括至少部分地由EPO生产缺陷（或低效）引起的疾病的管理，治疗和/或控制，相对于血红蛋白水平。

10. 发明申请

US20030187068A1 Substituted phenylpropionic acid derivatives 失效
标题翻译：取代苯基丙酸衍生物
公开(公告)号：US20030187068A1
公开(公告)日：2003-10-02
申请号：US10296206
申请日：2002-11-29
发明人： Hiroyuki Miyachi , Masahiro Nomura , Yukie Takahashi , Takahiro Tanase , Kouji Murakami , Masahiro Suzuki
IPC分类号： A61K031/195 , C07C235/52
CPC分类号： C07C229/34 , C07B2200/07 , C07C69/734 , C07C69/738 , C07C233/55 , C07C235/38
摘要： The invention provides novel substituted phenylpropionic acid derivatives that bind to the receptor as ligands of human peroxisome proliferator-activated receptor a (PPARnull) to activate and exhibit potent lipid-decreasing action, and processes for preparing them. It relates to substituted phenylpropionic acid derivatives represented by a general formula (1) 1 nullwherein R1 denotes a lower alkyl group with carbon atoms of 1 to 4, lower alkoxy group with carbon atoms of 1 to 3, trifluoromethyl group, trifluoromethoxy group, phenyl group which is unsubstituted or may have substituents, phenoxy group which is unsubstituted or may have substituents or benzyloxy group which is unsubstituted or may have substituents, R2 denotes a hydrogen atom, lower alkyl group with carbon atoms of 1 to 4 or lower alkoxy group with carbon atoms of 1 to 3, R3 denotes a lower alkoxy group with carbon atoms of 1 to 3, and the binding mode of A portion denotes nullCH2CONHnull, nullNHCOCH2null, nullCH2CH2COnull, nullCH2CH2CH2null, nullCH2CH2Onull, nullCONHCH2null, nullCH2NHCH2null, nullCOCH2Onull, nullOCH2COnull, nullCOCH2NHnull or nullCHCH2COnullnull, their pharmaceutically acceptable salts and their hydrates, and processes for preparing them.
摘要翻译：本发明提供新的取代的苯基丙酸衍生物，其结合受体作为人类过氧化物酶体增殖物激活受体α（PPARα）的配体，以激活并显示出有力的降脂作用，以及制备它们的方法。它涉及由通式（1）表示的取代的苯基丙酸衍生物[其中R 1表示碳原子数为1〜4的低级烷基，碳原子数1〜3的低级烷氧基，三氟甲基，三氟甲氧基，未取代或可具有取代基的苯基，未取代或可具有取代基的苯氧基或未取代或可具有取代基的苄氧基，R 2表示氢原子，碳原子数为1〜4的低级烷基或碳原子数为1〜3的低级烷氧基，R 3表示碳原子数为1〜3的低级烷氧基，A部分的结合方式表示-CH 2 CONH - ， - NHCOCH 2 - ， - CH 2 CH 2 CO-， - CH2CH2CH2-，-CH2CH2O-，-CONHCH2-，-CH2NHCH2-，-COCH2O-，-OCH2CO-，-COCH2NH-或-CHCH2CO-]，其药学上可接受的盐和它们的水合物，以及它们的制备方法。

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