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1. 发明申请

US20110309309A1 Oxocarbon-, Pseudooxocarbon- and Radialene Compounds and Their Use 有权
标题翻译：氧化碳，假氧化碳和镭二烯化合物及其用途
公开(公告)号：US20110309309A1
公开(公告)日：2011-12-22
申请号：US13178855
申请日：2011-07-08
申请人： Horst Hartmann , Olaf Zeika , Andrea Lux , Steffen Willmann
发明人： Horst Hartmann , Olaf Zeika , Andrea Lux , Steffen Willmann
IPC分类号： H01B1/12 , C07C255/31 , C07D409/14 , C07D333/22 , C07C49/603 , C07C13/19 , C07D401/14 , C07C49/297 , C07C49/303 , C07C13/04 , C07C13/11 , C07C49/293 , C07C255/50
CPC分类号： H01L51/005 , C07C13/04 , C07C13/06 , C07C13/11 , C07C13/19 , C07C49/39 , C07C49/395 , C07C49/653 , C07C255/31 , C07C255/40 , C07C255/51 , C07C261/04 , C07C325/02 , C07C2601/02 , C07C2601/04 , C07C2601/08 , C07C2601/14 , C07C2601/16 , C07D213/53 , C07D333/24 , C09B11/02 , C09B47/04 , C09B57/00 , C09B57/008 , H01L51/002 , H01L51/0051 , H01L51/0067 , H01L51/0068 , Y02E10/549 , Y02P70/521
摘要： The present invention relates to oxocarbon-, pseudooxocarbon- and radialene compounds as well as to their use as doping agent for doping an organic semiconductive matrix material, as blocker material, as charge injection layer, as electrode material as well as organic semiconductor, as well as electronic components and organic semiconductive materials using them.
摘要翻译：本发明涉及氧化碳 - 假氧化碳 - 和枞酸化合物，以及它们作为掺杂剂用作掺杂有机半导体基质材料作为阻挡剂材料，作为电荷注入层，作为电极材料以及有机半导体的用途，以及作为电子元件和使用它们的有机半导体材料。

2. 发明申请

US20050090562A1 Clusianon isomers and use thereof 失效
标题翻译： Clusianon异构体及其用途
公开(公告)号：US20050090562A1
公开(公告)日：2005-04-28
申请号：US10496592
申请日：2002-11-20
申请人： Siegfried Seeber , Ralf Hilger , David Diaz-Carballo
发明人： Siegfried Seeber , Ralf Hilger , David Diaz-Carballo
IPC分类号： A61P31/12 , A61K31/122 , A61K45/06 , A61P35/00 , A61P35/02 , A61P43/00 , C07C49/747 , C07C49/835 , C07C49/84 , A61K31/12 , C07C49/293
CPC分类号： C07C49/84 , A61K45/06 , C07C49/835
摘要： The invention relates to a clusianon isomer and to the use thereof, in particular as a pharmaceutical or medical active ingredient, in particular for producing medicaments for the prophylactic and/or therapeutic (curative) treatment of tumour or cancer diseases as well as viral diseases. The aforementioned compound can be used in cytostatics and antiviral agents (virostatics). Said compound acts, in particular, as a topoisomerase and telomerase inhibitor and as a regulator in the MAP kinase signal transduction. Said compound can thus intervene at the cellular level in the proliferation mechanism of tumour or cancer cells and viruses.
摘要翻译：本发明涉及克氏体异构体及其用途，特别是作为药物或医学活性成分，特别是用于生产用于预防和/或治疗（治疗）治疗肿瘤或癌症疾病以及病毒性疾病的药物。上述化合物可用于细胞抑制剂和抗病毒剂（静态）。所述化合物特别地作为拓扑异构酶和端粒酶抑制剂起作为MAP激酶信号转导中的调节剂的作用。因此，所述化合物可以在肿瘤或癌细胞和病毒的增殖机制中的细胞水平上干预。

3. 发明申请

US20050004385A1 Fulvene, metallocene catalysts and preparation method thereof, and preparation of polyolefines copolymer using the same 失效
标题翻译：呋喃，茂金属催化剂及其制备方法，以及使用其制备聚烯烃共聚物
公开(公告)号：US20050004385A1
公开(公告)日：2005-01-06
申请号：US10494213
申请日：2003-08-29
申请人： Young-Whan Park , Si-Geun Lee , Sung-Don Hong , Kwang-Ho Song , Boong-Goon Jeong , Dae-Woo Nam , Bun-Yeol Lee , Choong-hoon Lee , Hyo-Sun Lee
发明人： Young-Whan Park , Si-Geun Lee , Sung-Don Hong , Kwang-Ho Song , Boong-Goon Jeong , Dae-Woo Nam , Bun-Yeol Lee , Choong-hoon Lee , Hyo-Sun Lee
IPC分类号： C07D317/72 , C07C1/207 , C07C13/28 , C07C13/465 , C07C13/567 , C07C45/58 , C07C45/59 , C07C49/687 , C07C49/707 , C07C49/747 , C07C49/753 , C07F7/00 , C07F17/00 , C08F4/642 , C08F4/659 , C08F4/6592 , C08F4/76 , C08F10/00 , C08F110/02 , C08F210/02 , C07C49/293
CPC分类号： C07C45/59 , C07C45/58 , C07C49/687 , C07C49/707 , C07C49/747 , C07C49/753 , C08F4/65912 , C08F4/6592 , C08F110/02 , C08F210/02 , Y10S526/943 , C08F4/65927 , C08F232/00 , C08F2500/25 , C08F2500/03
摘要： The present invention relates to a novel fulvene compound and a preparation method thereof, and more particularly to a fulvene compound having substituted groups in the 2- and 5-positions, prepared from an unsaturated ketone having a substituted group in the β-position and a halogen atom in the α-position, and a preparation method thereof. The present invention also relates to a metallocene catalyst having a substituted group in the α-position carbon of the bridge of the cyclopentadienyl group only by reaction of a fulvene compound and an anion group including the cyclopentadienyl group, and a preparation method of a polyolefin copolymer using the same.
摘要翻译：本发明涉及一种新颖的富烯化合物及其制备方法，更具体地涉及由在β-位具有取代基的不饱和酮制备的2-和5-位具有取代基的富烯化合物和 α位的卤素原子及其制备方法。本发明还涉及仅通过富烯化合物和包括环戊二烯基的阴离子基团的反应在环戊二烯基桥的α位碳上具有取代基的茂金属催化剂，以及聚烯烃共聚物的制备方法使用相同

4. 发明授权

US5703246A Process for the preparation of an oxirane, azirdine or cyclopropane 失效
标题翻译：制备环氧乙烷，氮杂环丁烷或环丙烷的方法
公开(公告)号：US5703246A
公开(公告)日：1997-12-30
申请号：US617755
申请日：1996-03-15
申请人： Varinder Kumar Aggarwal , Hesham Nimer Hasan Abdel-Rahman , Hee Yoon Lee
发明人： Varinder Kumar Aggarwal , Hesham Nimer Hasan Abdel-Rahman , Hee Yoon Lee
IPC分类号： C07B37/10 , C07B41/00 , C07B43/00 , C07C2/86 , C07C13/04 , C07C13/28 , C07C45/68 , C07C49/293 , C07C69/743 , C07C69/753 , C07C211/16 , C07C303/30 , C07C303/34 , C07C303/40 , C07C315/04 , C07D203/02 , C07D203/22 , C07D203/24 , C07D301/02 , C07D303/04 , C07D303/08 , C07D303/16 , C07D303/40 , C07D303/46 , C07D407/04 , C07F9/564 , C07C203/00
CPC分类号： C07D203/22 , C07C2/868 , C07D203/02 , C07D203/24 , C07D301/02 , C07D303/04 , C07D303/08 , C07D303/16 , C07D303/40 , C07D303/46 , C07D407/04 , C07F9/564 , C07C2101/02
摘要： A process for the preparation of an oxirane, aziridine or cyclopropane of formula (I) wherein, X is oxygen, NR.sup.4 or CHR.sup.5 ; R.sup.1 is hydrogen, alkyl, aryl, heteroaromatic, heterocyclic or cycloalkyl; R.sup.2 is hydrogen, alkyl, aryl, heteroaromatic, CO.sub.2 R.sup.8, CHR.sup.14 NHR.sup.13, heterocyclic or cycloalkyl; or R.sup.1 and R.sup.2 join together to form a cycloalkyl ring; R.sup.3 is hydrogen, alkyl, aryl, heteroaromatic, CO.sub.2 R.sup.8, R.sup.8.sub.3 Sn, CONR.sup.8 R.sup.9 or trimethylsilyl; R.sup.4 and R.sup.5 are, independently, alkyl, cycloalkyl, aryl, heteroaromatic, SO.sub.2 R.sup.8, SO.sub.3 R.sup.8, COR.sup.8, CO.sub.2 R.sup.8, CONR.sup.8 R.sup.9 or CN, or R.sup.4 can also be P(O)(aryl).sub.2 ; R.sup.8 and R.sup.9 are independently alkyl, aryl or arylalkyl; R.sup.13 and R.sup.14 are independently hydrogen, alkyl or aryl; the process comprising reacting a mixture of a compound of formula (II), wherein R.sup.1, R.sup.2 and X are as defined above, and a sulphide of formula SR.sup.6 R.sup.7, wherein R.sup.6 and R.sup.7 are independently alkyl, aryl or heteroaomatic, or R.sup.6 and R.sup.7 join together to form a cycloalkyl ring which optionally includes an additional heteroatom, with either (i) a metallocarbon obtainable by reacting an alkylmetal with a methane derivative of formula CHR.sup.3 X'X", wherein R.sup.3 is as defined above, and X' and X" are independently, a leaving group, or (ii) a metallocarbon obtainable by reacting a compound of formula (III), (wherein R.sup.3 may not be hydrogen) with a suitable organometallic or inorganic reagent.
摘要翻译： PCT No.PCT / GB94 / 02280第 371日期：1996年3月15日 102（e）1996年3月15日PCT 1994年10月19日PCT PCT。公开号WO95 / 11230 日期：1995年04月27日制备式（I）的环氧乙烷，氮丙啶或环丙烷的方法，其中X是氧，NR 4或CHR 5; R 1是氢，烷基，芳基，杂芳族，杂环或环烷基; R2是氢，烷基，芳基，杂芳族，CO2R8，CHR14NHR13，杂环或环烷基; 或R 1和R 2连接在一起形成环烷基环; R3是氢，烷基，芳基，杂芳族，CO2R8，R83Sn，CONR8R9或三甲基甲硅烷基; R4和R5独立地是烷基，环烷基，芳基，杂芳族，SO2R8，SO3R8，COR8，CO2R8，CONR8R9或CN，或R4也可以是P（O）（芳基）2; R8和R9独立地是烷基，芳基或芳基烷基; R 13和R 14独立地是氢，烷基或芳基; 该方法包括使式（II）化合物（其中R 1，R 2和X如上所定义）和式SR 6 R 7的硫化物的混合物反应，其中R 6和R 7独立地为烷基，芳基或杂芳基，或R 6和R 7连接一起形成任选地包括另外的杂原子的环烷基环，与（i）通过使烷基金属与式CHR 3 X'X“的甲烷衍生物反应得到的金属碳，其中R 3如上所定义，X'和X' 独立地是离去基团，或（ii）可通过使式（III）化合物（其中R 3可以不是氢）与合适的有机金属或无机试剂反应得到的金属碳。

5. 发明授权

US4399163A Branched amides of L-aspartyl-D-amino acid dipeptides 失效
标题翻译： L-天冬氨酰-D-氨基酸二肽的分支酰胺
公开(公告)号：US4399163A
公开(公告)日：1983-08-16
申请号：US276243
申请日：1981-06-26
申请人： Thomas M. Brennan , Michael E. Hendrick
发明人： Thomas M. Brennan , Michael E. Hendrick
IPC分类号： A23L27/30 , C07C45/00 , C07C45/29 , C07C45/61 , C07C45/62 , C07C45/63 , C07C45/64 , C07C45/67 , C07C45/68 , C07C45/74 , C07C49/16 , C07C49/17 , C07C49/173 , C07C49/293 , C07C49/39 , C07C49/395 , C07C49/403 , C07C49/413 , C07C49/523 , C07C49/647 , C07C323/25 , C07D307/22 , C07D307/32 , C07D331/04 , C07D333/32 , C07D333/36 , C07D335/02 , C07K5/072 , C07K5/075 , A23L1/236
CPC分类号： C07D307/32 , A23L27/32 , C07C323/25 , C07C45/00 , C07C45/004 , C07C45/292 , C07C45/61 , C07C45/62 , C07C45/63 , C07C45/64 , C07C45/673 , C07C45/68 , C07C45/74 , C07C49/16 , C07C49/17 , C07C49/173 , C07C49/293 , C07C49/39 , C07C49/395 , C07C49/403 , C07C49/413 , C07C49/523 , C07C49/647 , C07D307/22 , C07D331/04 , C07D333/32 , C07D333/36 , C07D335/02 , C07K5/06113 , Y10S426/804 , Y10S530/801
摘要： Amides of L-aspartyl-D-amino acid dipeptides of the formula ##STR1## and physiologically acceptable cationic and acid addition salts thereof wherein R.sup.a is CH.sub.2 OH or CH.sub.2 OCH.sub.3 ; R is a branched member selected from the group consisting of fenchyl, diisopropylcarbinyl, d-methyl-t-butylcarbinyl, d-ethyl-t-butylcarbinyl, di-t-butyl-carbinyl, 2-methylthio-2,4-dimethylpentan-3-yl, ##STR2## said amides are potent sweeteners having advantages over the prior art, edible compositions containing them, methods for their use in edible compositions and novel amide intermediates useful in their production.
摘要翻译：式（I）的L-天冬氨酰-D-氨基酸二肽和其生理上可接受的阳离子和酸加成盐的酰胺，其中R a是CH 2 OH或CH 2 OCH 3; R是选自偕基，二异丙基脒基，二甲基 - 叔丁基carb基，二乙基 - 叔丁基咔inyl基，二 - 叔丁基 - 碳酰基，2-甲硫基-2,4-二甲基戊烷-3 所述酰胺是具有优于现有技术的有用甜味剂，含有它们的食用组合物，它们在食用组合物中的用途及其生产中可用的新型酰胺中间体。

6. 发明授权

US4154959A 11-(2-Hydroxyethylthio)prostenoic acid E series derivatives 失效
公开(公告)号：US4154959A
公开(公告)日：1979-05-15
申请号：US842844
申请日：1977-10-17
申请人： Martin J. Weiss , Gerald J. Siuta
发明人： Martin J. Weiss , Gerald J. Siuta
IPC分类号： C07C29/09 , C07C29/10 , C07C29/40 , C07C29/42 , C07C29/62 , C07C31/133 , C07C35/06 , C07C45/45 , C07C49/293 , C07C405/00 , C07F7/08 , C07F7/18 , C07F7/22 , C07C177/00
CPC分类号： C07F7/2212 , C07C29/095 , C07C29/10 , C07C29/40 , C07C29/42 , C07C29/62 , C07C31/1336 , C07C35/06 , C07C405/0033 , C07F7/0812 , C07F7/0818 , C07F7/1804 , C07B2200/07 , C07B2200/09 , C07C2101/02 , C07C2101/04 , C07C2101/08 , C07C2101/14 , Y10T83/8858
摘要： This disclosure describes certain 11-(2-hydroxyethylthio)-9-keto-prostenoic acid E series derivatives, and their intermediates, useful as bronchodilators and inflammatory medeator release inhibitors.

7. 发明授权

US5629455A Process for preparing cyclopropyl alkyl ketones and 4,5-dihydroalkylfurans 失效
标题翻译：制备环丙基烷基酮和4,5-二氢烷基呋喃的方法
公开(公告)号：US5629455A
公开(公告)日：1997-05-13
申请号：US589952
申请日：1996-01-23
申请人： Manfred Kaufhold , Marcel Feld
发明人： Manfred Kaufhold , Marcel Feld
IPC分类号： C07C45/59 , C07C45/67 , C07C49/293 , C07C49/317 , C07C49/792 , C07D307/28 , C07C45/54
CPC分类号： C07D307/28 , C07C45/676
摘要： The invention relates to a novel process for the simultaneous preparation of cyclopropyl alkyl ketones and 4,5-dihydroalkylfurans from 3-acyltetrahydrofuran-2-ones using a metal salt according to the diagram ##STR1## In the reaction, N-alkyllactams and/or N-acylmorpholines which are high-boiling and only slightly miscible with water are used. By charging the solvent, the metal salt and the 3-acyltetrahydrofuran-2-one in a molar excess with respect to the metal salt, heating the mixture to 160.degree. to 220.degree. C. and metering in further 3-acyl-tetrahydrofuran-2-one, the desired products are obtained in high yields. The metal salt can moreover be recovered in a simple manner by washing with water.
摘要翻译：本发明涉及一种根据图中使用金属盐从3-酰基四氢呋喃-2-酮同时制备环丙基烷基酮和4,5-二氢烷基呋喃的新方法。在反应中，N - 烷基内酰胺和/或N-酰基吗啉，它们是高沸点且仅与水轻微混溶。通过将溶剂，金属盐和3-酰基四氢呋喃-2-酮相对于金属盐摩尔过量地加入，将混合物加热至160℃至220℃，并进一步计量3-酰基 - 四氢呋喃-2 - 一种，以高产率获得所需的产物。此外，金属盐可以通过用水洗涤以简单的方式回收。

8. 发明授权

US5151447A S-substituted beta-thioacrylamide biocides and fungicides 失效
标题翻译： S-取代的β-硫代丙烯酰胺杀生物剂和杀真菌剂
公开(公告)号：US5151447A
公开(公告)日：1992-09-29
申请号：US533566
申请日：1990-06-05
申请人： David R. Amick
发明人： David R. Amick
IPC分类号： A01N37/36 , A01N37/42 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/78 , C07C45/45 , C07C49/293 , C07C323/60 , C07D275/02 , C07D275/03
CPC分类号： C07D275/03 , A01N37/36 , A01N37/42 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/78 , C07C323/60 , C07C45/455 , C07C49/293
摘要： S-substituted beta-thioacrylamide compounds have been discovered to be useful as biocides and fungicides. Compositions comprising the compound and isothiazolin-3-ones and/or carriers, methods of preparation of the compounds and methods of using the compounds and compositions are also disclosed.
摘要翻译：已经发现S-取代的β-硫代丙烯酰胺化合物可用作杀生物剂和杀真菌剂。还公开了包含化合物和异噻唑啉-3-酮和/或载体的组合物，化合物的制备方法和使用该化合物和组合物的方法。

9. 发明授权

US4983208A Fungicidal and plant growth-regulating hydroxyalkylazolyl derivatives 失效
标题翻译：杀真菌和植物生长调节羟烷基唑衍生物
公开(公告)号：US4983208A
公开(公告)日：1991-01-08
申请号：US406996
申请日：1989-09-14
申请人： Klaus Stroech , Monika Frie , Thomas Himmler , Wilhelm Brandes , Stefan Dutzmann , Gerd Hanssler
发明人： Klaus Stroech , Monika Frie , Thomas Himmler , Wilhelm Brandes , Stefan Dutzmann , Gerd Hanssler
IPC分类号： A01N31/04 , A01N31/14 , A01N43/32 , A01N43/50 , A01N43/653 , C07C33/50 , C07C45/62 , C07C45/74 , C07C49/163 , C07C49/225 , C07C49/237 , C07C49/293 , C07C49/327 , C07C49/457 , C07C49/467 , C07C49/533 , C07C49/563 , C07C49/567 , C07C49/657 , C07C49/687 , C07C49/693 , C07C49/753 , C07C317/24 , C07C323/22 , C07D20060101 , C07D233/60 , C07D233/61 , C07D249/08 , C07D303/08 , C07D303/22 , C07D303/34 , C07D319/16 , C07D319/18 , C07D319/20 , C07D405/06 , C07D407/06 , C07D521/00
CPC分类号： C07D303/22 , A01N43/653 , C07C321/00 , C07C33/50 , C07C45/62 , C07C45/74 , C07C49/457 , C07C49/467 , C07C49/567 , C07C49/657 , C07C49/687 , C07C49/693 , C07C49/753 , C07D231/12 , C07D233/56 , C07D249/08 , C07D303/08 , C07D303/34 , C07D407/06
摘要： Fungicidal and plant growth-regulating hydroxyalkylazolyl derivatives of the formula ##STR1## in which R represents hydrogen, alkyl or acyl,R.sup.1 represents halogen, optionally substituted phenyl or the grouping --Z--R.sup.3, whereinZ represents oxygen, sulphur, SO or SO.sub.2 andR.sup.3 represents optionally substituted alkyl, optionally substituted phenyl or optionally substituted phenylalkyl,R.sup.2 represents optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted naphthyl or the radical of the formula ##STR2## m represents the numbers, 0, 1, 2 or 3, or R.sup.2 represents the radical or the formula ##STR3## X represents nitrogen or a CH group and Y represents the groupings --CH.sub.2 --CH.sub.2 --, --CH.dbd.CH--, --C.tbd.C--, ##STR4## and their addition products with acids and metal salts. Intermediates of the formulas ##STR5## are also new.

10. 发明授权

US4833157A Methods of inhibitng gastric secretion with prostaglandin derivatives 失效
标题翻译：用前列腺素衍生物抑制胃分泌的方法
公开(公告)号：US4833157A
公开(公告)日：1989-05-23
申请号：US140729
申请日：1988-01-04
申请人： Harold C. Kluender , Warren D. Woessner , William G. Biddlecom
发明人： Harold C. Kluender , Warren D. Woessner , William G. Biddlecom
IPC分类号： C07C29/09 , C07C29/147 , C07C29/36 , C07C29/42 , C07C29/62 , C07C45/30 , C07C45/45 , C07C45/62 , C07C47/293 , C07C47/30 , C07C49/293 , C07C49/433 , C07C49/443 , C07C51/09 , C07C51/353 , C07C51/38 , C07C61/04 , C07C61/08 , C07C405/00 , C07F1/08
CPC分类号： C07F1/08 , C07C29/095 , C07C29/147 , C07C29/36 , C07C29/42 , C07C29/62 , C07C405/00 , C07C405/0025 , C07C45/305 , C07C45/45 , C07C45/62 , C07C47/293 , C07C47/30 , C07C49/293 , C07C49/433 , C07C49/443 , C07C51/09 , C07C51/353 , C07C51/38 , C07C61/04 , C07C61/08 , C07B2200/07 , C07B2200/09 , C07C2101/04 , C07C2101/08 , C07C2101/14 , C07C2102/20 , C07C2102/22 , Y10S514/926 , Y10S514/927
摘要： A therapeutic method for inhibiting gastric secretion in an individual for whom such therapy is indicated is disclosed. The method comprises administering to such an individual an effective inhibitory amount of certain derivatives of 15-deoxy-16-hydroxy-prostaglandin E.sub.1 esters.
摘要翻译：公开了一种治疗方法，用于抑制表达这种治疗的个体中的胃分泌。该方法包括向这样的个体施用有效抑制量的15-脱氧-16-羟基 - 前列腺素E1酯的某些衍生物。

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